SCHEMBL4742618

SCHEMBL4742618

O=C(CC(NC(=O)c1cnc2c([N+](=O)[O-])cccc2c1N1CCNCC1)C(=O)CF)OC(=O)C(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.34
TP53 P04637 1/20 0.34
MAPK1 P28482 1/20 0.34
RECQL P46063 1/20 0.34
HSD17B10 Q99714 1/20 0.34
MAPT P10636 4/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
MET P08581 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
MITF O75030 1/20 0.31
HTT P42858 1/20 0.31
HTR6 P50406 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4739351 0.91 MAPK1 (0.35) USP2TP53MAPK1RECQLHSD17B10
SCHEMBL4742160 0.90 MEN1 (0.36) USP2TP53MAPK1RECQLHSD17B10
SCHEMBL4743039 0.90 USP2 (0.35) USP2TP53MAPK1RECQLHSD17B10
SCHEMBL4742574 0.88 DRD2 (0.35) USP2TP53MAPK1RECQLHSD17B10
SCHEMBL4742118 0.85 MET (0.38) RECQLMAPTMEN1KMT2AMET
Trifluoroacetic Acid SCHEMBL4739344 0.81 SIRT6 (0.36) USP2TP53MAPK1RECQLHSD17B10
SCHEMBL4739340 0.81 THRB (0.40)
SCHEMBL4742120 0.81 THRB (0.43) MET
Trifluoroacetic Acid SCHEMBL4742157 0.80 MEN1 (0.36) USP2TP53MAPK1RECQLHSD17B10
SCHEMBL4743406 0.80 MET (0.39) USP2TP53MAPK1RECQLHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008093940-A1 QUINOLINE DERIVATIVES AS CASPASE-3 INHIBITOR, PREPARATION PROCESS FOR THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME YUNGJIN PHARMACEUTICAL CO., LTD. (KR) 2008-08-07 WO claimed
WO-2008093940-A1 QUINOLINE DERIVATIVES AS CASPASE-3 INHIBITOR, PREPARATION PROCESS FOR THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME YUNGJIN PHARMACEUTICAL CO., LTD. (KR) 2008-08-07 WO disclosed