SCHEMBL4748846

SCHEMBL4748846

Cc1cc(Oc2c[nH]nc2C2CC2)ccc1C#N

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESRRA P11474 1/20 0.41
AR P10275 10/20 0.40
SLC22A12 Q96S37 2/20 0.38
CYP19A1 P11511 1/20 0.35
MRGPRX4 Q96LA9 1/20 0.35
BCAT1 P54687 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4103776 0.83 PKM (0.34) SLC22A12
SCHEMBL4751336 0.79 RAPGEF4 (0.34) SLC22A12
SCHEMBL4751277 0.78 AR (0.40) ESRRAARSLC22A12MRGPRX4BCAT1
SCHEMBL4105432 0.78 AR (0.38) ESRRAARSLC22A12MRGPRX4
SCHEMBL4109832 0.74 ENPP3 (0.39) ESRRAARSLC22A12
SCHEMBL4751257 0.71 P2RY12 (0.37) ARMRGPRX4NPC1RAB9A
SCHEMBL17156280 0.70 HTR1A (0.45) CYP19A1
SCHEMBL16635898 0.70 KDM4E (0.32)
SCHEMBL13890508 0.69 AR (0.66) ARSLC22A12CYP19A1
SCHEMBL17645458 0.69 TGFBR1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008135824-A1 OXYALKYLPYRAZOLE COMPOUNDS USEFUL IN THERAPY PFIZER LIMITED (GB) 2008-11-13 WO disclosed