SCHEMBL4748849

SCHEMBL4748849

Cc1cc(OC(C=O)C2CC2)ccc1C#N

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.43
MRGPRX4 Q96LA9 1/20 0.39
ESRRA P11474 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
USP30 Q70CQ3 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
S1PR1 P21453 3/20 0.34
S1PR5 Q9H228 3/20 0.34
S1PR3 Q99500 2/20 0.33
DPP4 P27487 1/20 0.33
KCNH2 Q12809 1/20 0.33
PLA2G7 Q13093 1/20 0.33
CYP11B2 P19099 1/20 0.33
XDH P47989 1/20 0.33
S1PR4 O95977 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4751606 0.84 PGR (0.44) ARMRGPRX4ESRRA
SCHEMBL24074650 0.79 AR (0.46) ARMRGPRX4TDP1CYP11B2XDH
SCHEMBL4751285 0.77 ALDH1A1 (0.32) DPP4KCNH2
SCHEMBL28338571 0.71 AR (0.45) ARMRGPRX4ESRRAUSP30S1PR3
SCHEMBL18621197 0.71 AR (0.45) ARMRGPRX4S1PR3
SCHEMBL16483388 0.68 AR (0.48) ARMRGPRX4
SCHEMBL14022463 0.68 RAB9A (0.65) ARMRGPRX4NPC1RAB9AUSP30
SCHEMBL21237872 0.68 ATM (0.53) ARMRGPRX4NPC1RAB9ATDP1
SCHEMBL509379 0.67 AR (0.50) ARMRGPRX4NPC1RAB9A
SCHEMBL14553122 0.67 AR (0.47) ARMRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008135824-A1 OXYALKYLPYRAZOLE COMPOUNDS USEFUL IN THERAPY PFIZER LIMITED (GB) 2008-11-13 WO disclosed