SCHEMBL4752402

SCHEMBL4752402

CC(=O)OC1CN(Cc2ccccc2)CCN1Cc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.51
BCHE P06276 2/20 0.46
CYP2D6 P10635 1/20 0.46
LMNA P02545 1/20 0.46
POLB P06746 1/20 0.46
MAOB P27338 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27801284 0.87 SIGMAR1 (0.49) SIGMAR1BCHELMNAMAOB
SCHEMBL691442 0.86 BCHE (0.46) SIGMAR1BCHEMAOB
SCHEMBL27765696 0.81 SIGMAR1 (0.56) SIGMAR1LMNAPOLB
SCHEMBL4812815 0.79 AGTR2 (0.43) BCHE
SCHEMBL2628898 0.79 AGTR2 (0.52) SIGMAR1LMNA
SCHEMBL3206960 0.78 BCHE (0.60) BCHEMAOB
SCHEMBL9685669 0.78 BCHE (0.60) BCHEMAOB
SCHEMBL2893650 0.78 BCHE (0.60) BCHEMAOB
SCHEMBL9818951 0.77 BCHE (0.44) BCHEPOLB
SCHEMBL18498897 0.77 S1PR5 (0.53) BCHEMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008139941-A1 SUBSTITUTED IMIDAZOLE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-11-20 WO disclosed
EP-1984355-A2 CYCLIC AMINE COMPOUND AND USE THEREOF FOR THE PROPHYLAXIS OR TREATMENT OF HYPERTENSION Takeda Pharmaceutical Company Limited (JP) 2008-10-29 EP disclosed
WO-2007094513-A2 CYCLIC AMINE COMPOUND AND USE THEREOF FOR THE PROPHYLAXIS OR TREATMENT OF HYPERTENSION TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-08-23 WO disclosed