SCHEMBL4752969

SCHEMBL4752969

CC1(C)Cc2cc(S(=O)(=O)Nc3ccc(Cl)c(Cl)c3)cc(O)c2O1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PKM P14618 6/20 0.46
PKLR P30613 1/20 0.46
HSD17B3 P37058 1/20 0.42
HSD17B2 P37059 1/20 0.42
CYP26A1 O43174 1/20 0.41
CYP26B1 Q9NR63 1/20 0.41
MAPT P10636 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
CDK1 P06493 1/20 0.39
CCNB1 P14635 1/20 0.39
CCNA2 P20248 1/20 0.39
CDK2 P24941 1/20 0.39
CDK7 P50613 1/20 0.39
CCNH P51946 1/20 0.39
CCNA1 P78396 1/20 0.39
THRB P10828 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HTR6 P50406 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4752457 0.83 PKM (0.41) PKMPKLRCYP26A1CYP26B1THRB
SCHEMBL4754001 0.81 PKM (0.41) PKMPKLRCYP26A1CYP26B1MAPT
SCHEMBL4788883 0.78 TSHR (0.39) PKMCYP26A1CYP26B1MAPTALDH1A1
SCHEMBL4787216 0.74 AKT1 (0.38) MAPTALDH1A1
SCHEMBL4868478 0.70 LMNA (0.42) PKMMAPTALDH1A1NPSR1
SCHEMBL4750485 0.68 HTR2A (0.51) PKMALDH1A1NPSR1
SCHEMBL10361762 0.67 MAPT (0.65) PKMPKLRHSD17B3HSD17B2MAPT
SCHEMBL31589145 0.67 CDK1 (0.60) PKMPKLRHSD17B3HSD17B2MAPT
SCHEMBL7571133 0.65 MAPT (0.63) MAPTTDP1CDK1CCNB1CCNA2
SCHEMBL7563643 0.65 CES1 (0.72) HSD17B3HSD17B2MAPTTDP1CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008146064-A1 NEW BENZOFURAN DERIVATIVES AS SELECTIVE 5HT7 RECEPTOR INHIBITORS AND PROCESS FOR THEIR PREPARATION EGIS GYÓGYSZERGYÁR (HU) 2008-12-04 WO disclosed