SCHEMBL4753718

SCHEMBL4753718

O=C(O)c1cc(=O)nc([C@H]2CC[C@@H](C(F)(F)F)CC2)n1-c1ccc(Cl)nc1

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 1/20 0.33
AKR1C3 P42330 1/20 0.32
CHRM4 P08173 2/20 0.32
LPL P06858 1/20 0.32
LIPG Q9Y5X9 1/20 0.32
GRM5 P41594 1/20 0.32
PIK3CA P42336 2/20 0.32
AVPR1A P37288 1/20 0.32
PDE4B Q07343 1/20 0.31
PDE4D Q08499 1/20 0.31
CHRNB2 P17787 3/20 0.31
CHRNA4 P43681 3/20 0.31
NAPRT Q6XQN6 1/20 0.31
USP14 P54578 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
RHOA P61586 1/20 0.30
CHRNB4 P30926 1/20 0.30
CHRNA3 P32297 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4755067 0.88 AVPR1A (0.37) TBK1GRM5AVPR1APDE4BKDM4E
SCHEMBL13985224 0.84 TBK1 (0.33) TBK1AKR1C3CHRM4LPLLIPG
SCHEMBL4755767 0.78 CHRNB2 (0.34) PIK3CAAVPR1ACHRNB2CHRNA4USP14
SCHEMBL4755765 0.78 CHRNB2 (0.34) PIK3CAAVPR1ACHRNB2CHRNA4USP14
SCHEMBL4755763 0.75 PIK3CA (0.36) CHRM4PIK3CAAVPR1ACHRNB2CHRNA4
SCHEMBL4755760 0.75 PIK3CA (0.36) CHRM4PIK3CAAVPR1ACHRNB2CHRNA4
SCHEMBL3174423 0.73 PDE4B (0.36) PDE4BPDE4DCHRNB2CHRNA4USP14
SCHEMBL3174425 0.73 PDE4B (0.36) PDE4BPDE4DCHRNB2CHRNA4USP14
SCHEMBL13985414 0.73 DGAT1 (0.33)
SCHEMBL3169414 0.71 YTHDC1 (0.35) PIK3CAPDE4BPDE4DCHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008156607-A1 SUBSTITUTED PYRIMIDINONES NEUROGEN CORPORATION (US) 2008-12-24 WO disclosed