SCHEMBL4755368

SCHEMBL4755368

CC1=C(C(=O)O)C(c2ccccc2F)(C(C)(C)C)C(C(=O)O)=C(C)N1C(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.36
HDAC4 P56524 9/20 0.35
NOTUM Q6P988 2/20 0.33
OPRL1 P41146 2/20 0.33
HDAC9 Q9UKV0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4757278 0.72 CYP2C9 (0.34) NOTUM
SCHEMBL4755316 0.65 HCAR2 (0.36) HCAR2HDAC4NOTUM
SCHEMBL9505359 0.61 KDM4E (0.49)
SCHEMBL7776061 0.60 CRHBP (0.43) HCAR2HDAC4OPRL1
SCHEMBL803450 0.57 HDAC4 (0.40) HCAR2HDAC4OPRL1
SCHEMBL20249893 0.57 THRB (0.46) HCAR2HDAC4OPRL1HDAC9
SCHEMBL31125559 0.56 HDAC4 (0.59) HCAR2HDAC4OPRL1
SCHEMBL301133 0.56 HDAC4 (0.59) HCAR2HDAC4OPRL1
Acetic Acid SCHEMBL27477632 0.56 CES2 (0.52)
SCHEMBL29177458 0.55 OPRM1 (0.44) HCAR2HDAC4NOTUMOPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008006070-A2 COMPOUNDS AND COMBINATIONS THEREOF FOR INHIBITING BETA-AMYLOID PRODUCTION AND METHODS OF USE THEREOF ROSKAMP RESEARCH LLC (US) 2008-01-10 WO disclosed
EP-1858325-A2 COMPOUNDS FOR INHIBITING BETA-AMYLOID PRODUCTION AND METHODS OF IDENTIFYING THE COMPOUNDS Roskamp Research LLC (US) 2007-11-28 EP disclosed
WO-2006074419-A2 COMPOUNDS FOR INHIBITING BETA-AMYLOID PRODUCTION AND METHODS OF IDENTIFYING THE COMPOUNDS ROSKAMP RESEARCH LLC (US) 2006-07-13 WO disclosed