SCHEMBL4756534

SCHEMBL4756534

CNc1c(Cl)c(=O)nc([C@H]2CC[C@@H](C(F)(F)F)CC2)n1-c1ccc(C(N)=O)nc1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KIT P10721 6/20 0.34
FLT3 P36888 6/20 0.34
KMT2A Q03164 1/20 0.32
PARP1 P09874 5/20 0.32
HTR2A P28223 1/20 0.32
HRH3 Q9Y5N1 3/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
PARP2 Q9UGN5 3/20 0.32
PARP6 Q2NL67 2/20 0.32
PARP3 Q9Y6F1 2/20 0.32
TNKS O95271 2/20 0.31
GRM2 Q14416 1/20 0.31
PI4KB Q9UBF8 1/20 0.31
LRRK2 Q5S007 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4755127 0.83 PDE4B (0.35) LRRK2KCNH2
SCHEMBL4756663 0.79 RORC (0.35) KCNH2
SCHEMBL4755763 0.72 PIK3CA (0.36) LRRK2
SCHEMBL4755760 0.72 PIK3CA (0.36) LRRK2
SCHEMBL4755548 0.70 PDE4B (0.35) LRRK2
SCHEMBL4755555 0.70 PDE4B (0.35) LRRK2
SCHEMBL13985224 0.68 TBK1 (0.33)
SCHEMBL4755228 0.68 DRD1 (0.40) KMT2AKDM4EMAPTKCNH2
SCHEMBL4755225 0.68 DRD1 (0.40) KMT2AKDM4EMAPTKCNH2
SCHEMBL4756551 0.68 DRD1 (0.40) KMT2AKDM4EMAPTKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008156607-A1 SUBSTITUTED PYRIMIDINONES NEUROGEN CORPORATION (US) 2008-12-24 WO claimed