SCHEMBL4756663

SCHEMBL4756663

CNc1c(Cl)c(=O)nc([C@H]2CC[C@@H](C(F)(F)F)CC2)n1-c1ccc(C#N)cc1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RORC P51449 3/20 0.35
HSD11B1 P28845 1/20 0.35
CXCR3 P49682 3/20 0.33
AVPR1A P37288 1/20 0.32
USP14 P54578 6/20 0.32
CRHR1 P34998 1/20 0.31
PDE4B Q07343 1/20 0.31
DRD2 P14416 2/20 0.30
DRD4 P21917 2/20 0.30
DRD3 P35462 2/20 0.30
KCNH2 Q12809 1/20 0.30
CYP11B2 P19099 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4755127 0.87 PDE4B (0.35) USP14PDE4BDRD2DRD3KCNH2
SCHEMBL13985527 0.81 HSD11B1 (0.36) RORCHSD11B1CXCR3AVPR1AUSP14
SCHEMBL13985228 0.79 CRHR1 (0.35) RORCHSD11B1AVPR1AUSP14CRHR1
SCHEMBL4756580 0.79 USP14 (0.36) HSD11B1AVPR1AUSP14CRHR1
SCHEMBL4756534 0.79 KIT (0.34) KCNH2
SCHEMBL13985417 0.76 HSD11B1 (0.37) HSD11B1AVPR1AUSP14CRHR1DRD2
SCHEMBL13985520 0.76 USP14 (0.38) HSD11B1AVPR1AUSP14DRD2DRD4
SCHEMBL4755555 0.73 PDE4B (0.35) USP14PDE4B
SCHEMBL4755548 0.73 PDE4B (0.35) USP14PDE4B
SCHEMBL4755228 0.73 DRD1 (0.40) RORCAVPR1ACRHR1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008156607-A1 SUBSTITUTED PYRIMIDINONES NEUROGEN CORPORATION (US) 2008-12-24 WO claimed