SCHEMBL4757375

SCHEMBL4757375

CNCc1[c]c(-c2ccccc2)ccc1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.45
CYP3A4 P08684 1/20 0.45
MAPT P10636 1/20 0.45
PRMT6 Q96LA8 7/20 0.38
HTR7 P34969 1/20 0.37
EPHX2 P34913 1/20 0.36
CD274 Q9NZQ7 2/20 0.33
IFNAR1 P17181 1/20 0.33
SOS1 Q07889 1/20 0.32
ATM Q13315 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31
HTR2A P28223 1/20 0.31
SLC6A4 P31645 1/20 0.31
CARM1 Q86X55 1/20 0.31
NOS1 P29475 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6286439 0.79 TP53 (0.36) MAPTTAAR1
SCHEMBL17697662 0.77 CALM1 (0.42) KDM4ECYP3A4MAPTTAAR1
SCHEMBL7311782 0.75 ALDH1A1 (0.36) TAAR1
SCHEMBL28033340 0.75 TAAR1 (0.45) CYP3A4TAAR1
SCHEMBL27651823 0.72 KDM4E (0.37) KDM4ECYP3A4MAPTPRMT6IFNAR1
SCHEMBL379055 0.72 ALDH1A1 (0.47) CYP3A4MAPTATMTAAR1SLC6A4
SCHEMBL21177097 0.71 KDM4E (0.35) KDM4ECYP3A4MAPTPRMT6IFNAR1
SCHEMBL15756039 0.70 GABRA1 (0.35)
SCHEMBL27472235 0.70
SCHEMBL7307513 0.68 CYP2D6 (0.35) KDM4ECYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008124575-A1 RENIN INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-10-16 WO disclosed