SCHEMBL4758256

SCHEMBL4758256

CCOC(=O)c1cc(Cl)cc(C2=CCNCC2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 4/20 0.46
SIGMAR1 Q99720 2/20 0.44
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
HTR6 P50406 6/20 0.41
FTO Q9C0B1 1/20 0.39
MAPT P10636 1/20 0.39
HTR1B P28222 1/20 0.39
HTR2A P28223 1/20 0.39
HTR7 P34969 1/20 0.39
HTR3A P46098 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
QDPR P09417 3/20 0.39
CCNT1 O60563 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13944380 0.82 QDPR (0.51) HTR2CSIGMAR1SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL4185793 0.81 QDPR (0.50) HTR2CSIGMAR1SLC6A2SLC6A4SLC6A3
SCHEMBL28688462 0.75 SIGMAR1 (0.69) HTR2CSIGMAR1HTR6MAPTHTR1B
Hydrochloric Acid SCHEMBL28678896 0.73 HTR2C (0.70) HTR2CSIGMAR1HTR6FTOMAPT
SCHEMBL2662880 0.73 CA12 (0.62) CA12CA1CA2CA7CA9
SCHEMBL7589274 0.73 CA12 (0.62) CA12CA1CA2CA7CA9
SCHEMBL4756934 0.72 PPARG (0.44) SIGMAR1MAPT
SCHEMBL4757771 0.71 PDK4 (0.45)
SCHEMBL15787045 0.71 IMPDH2 (0.58) HTR2CHTR6MAPT
SCHEMBL4869840 0.71 TSHR (0.56) SLC6A2SLC6A4SLC6A3MAPTCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009000819-A1 5-PHENYL-1,3,4-OXADIAZOL-2-YL-ACETYL-4-PIPERIDINYL DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2008-12-31 WO disclosed
WO-2009000819-A1 5-PHENYL-1,3,4-OXADIAZOL-2-YL-ACETYL-4-PIPERIDINYL DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2008-12-31 WO disclosed