SCHEMBL4759543

SCHEMBL4759543

CCCCOC(=O)NC(Cc1cc(C)n(C)n1)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 9/20 0.40
ITGA2B P08514 8/20 0.40
ALDH1A1 P00352 3/20 0.39
CYP3A4 P08684 2/20 0.39
HPGD P15428 1/20 0.39
ACE P12821 2/20 0.39
ACE2 Q9BYF1 2/20 0.39
ITGB1 P05556 1/20 0.39
ITGA4 P13612 1/20 0.39
CPB2 Q96IY4 1/20 0.38
MAPK1 P28482 2/20 0.37
TSHR P16473 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MAPT P10636 1/20 0.37
GLA P06280 1/20 0.36
KMT2A Q03164 1/20 0.36
ITGAV P06756 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1196352 0.80 ACE (0.48) ITGB3ITGA2BALDH1A1CYP3A4HPGD
SCHEMBL1196353 0.80 ACE (0.48) ITGB3ITGA2BALDH1A1CYP3A4HPGD
SCHEMBL5500074 0.78 CPB2 (0.47) ITGB3ITGA2BACEACE2CPB2
SCHEMBL7300962 0.78 ITGB3 (0.41) ITGB3ITGA2BACEACE2ITGB1
SCHEMBL7300949 0.78 ITGB3 (0.41) ITGB3ITGA2BACEACE2ITGB1
SCHEMBL4759546 0.75 SMN1; SMN2 (0.37) ALDH1A1HPGDMAPK1TSHRL3MBTL1
SCHEMBL3663113 0.74 CTSK (0.47) ITGB3ITGA2BACEACE2ITGB1
SCHEMBL5086307 0.74 HDAC6 (0.49) ITGB3ITGA2BHPGDACEACE2
SCHEMBL10477488 0.74 ITGB1 (0.43) ITGB3ITGA2BHPGDITGB1ITGA4
SCHEMBL6015436 0.74 ITGB1 (0.43) ITGB3ITGA2BHPGDITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981854-A1 ARYLPROPIONAMIDE, ARYLACRYLAMIDE, ARYLPROPYNAMIDE, OR ARYLMETHYLUREA ANALOGS AS FACTOR XIA INHIBITORS Brystol-Myers Squibb Company (US) 2008-10-22 EP disclosed
WO-2007070826-A1 ARYLPROPIONAMIDE, ARYLACRYLAMIDE, ARYLPROPYNAMIDE, OR ARYLMETHYLUREA ANALOGS AS FACTOR XIA INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-06-21 WO disclosed