SCHEMBL4775781

SCHEMBL4775781

Cc1ccc(S(=O)(=O)Nc2ccc(O)cc2-c2ncco2)cc1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
MCOLN3 Q8TDD5 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
PIK3CD O00329 1/20 0.45
PIK3CG P48736 1/20 0.45
LMNA P02545 2/20 0.39
HTT P42858 2/20 0.39
GAA P10253 1/20 0.39
PKM P14618 1/20 0.39
POLB P06746 1/20 0.39
CYTH2 Q99418 2/20 0.38
RET P07949 2/20 0.38
RIPK2 O43353 1/20 0.38
KDR P35968 1/20 0.38
MAPK14 Q16539 1/20 0.38
PKMYT1 Q99640 1/20 0.38
KDM4E B2RXH2 1/20 0.37
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4780645 0.90 PIK3CD (0.43) ALDH1A1MCOLN3L3MBTL1PIK3CDPIK3CG
SCHEMBL4781338 0.86 SLC40A1 (0.48) ALDH1A1LMNAHTTGAAKDM4E
SCHEMBL4777554 0.85 PKM (0.46) ALDH1A1MCOLN3L3MBTL1PIK3CDPIK3CG
SCHEMBL4781354 0.82 BRAF (0.42) POLBKDRMEN1KMT2ACCR2
SCHEMBL4780299 0.81 CYP3A4 (0.41) ALDH1A1LMNAPKMPOLBMEN1
SCHEMBL3091703 0.81 CCR9 (0.43) PIK3CDPIK3CGGAAMEN1KMT2A
SCHEMBL4780017 0.81 KAT6A (0.39) ALDH1A1PIK3CDPIK3CGHTTGAA
SCHEMBL4779280 0.79 SLC40A1 (0.51) LMNAGAATSHRMEN1KMT2A
SCHEMBL4781379 0.76 TSHR (0.46) ALDH1A1LMNAHTTKDM4ETSHR
SCHEMBL4781517 0.73 MEN1 (0.41) POLBKDRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008008374-A2 CCR2 INHIBITORS AND METHODS OF USE THEREOF CHEMOCENTRYX, INC. (US) 2008-01-17 WO claimed
WO-2008008374-A2 CCR2 INHIBITORS AND METHODS OF USE THEREOF CHEMOCENTRYX, INC. (US) 2008-01-17 WO disclosed