SCHEMBL4777554

SCHEMBL4777554

COc1ccc(NS(=O)(=O)c2ccc(C)c(C)c2)c(-c2ncco2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.46
FFAR4 Q5NUL3 2/20 0.46
ALDH1A1 P00352 5/20 0.45
LMNA P02545 3/20 0.45
HTT P42858 3/20 0.45
MCOLN3 Q8TDD5 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
KDM4E B2RXH2 1/20 0.44
CCR9 P51686 1/20 0.43
KMT2A Q03164 4/20 0.43
MEN1 O00255 3/20 0.43
GAA P10253 1/20 0.43
TSHR P16473 3/20 0.42
KEAP1 Q14145 3/20 0.42
NPSR1 Q6W5P4 2/20 0.42
NFE2L2 Q16236 2/20 0.42
PIK3CD O00329 1/20 0.42
PIK3CG P48736 1/20 0.42
POLB P06746 1/20 0.42
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4781379 0.91 TSHR (0.46) FFAR4ALDH1A1LMNAHTTKDM4E
SCHEMBL3095654 0.86 STAT3 (0.51) ALDH1A1LMNAHTTKDM4ECCR9
SCHEMBL30304671 0.86 KEAP1 (0.50) LMNAHTTCCR9KMT2AMEN1
SCHEMBL18315257 0.86 KEAP1 (0.50) LMNAHTTCCR9KMT2AMEN1
SCHEMBL4775781 0.85 ALDH1A1 (0.46) PKMALDH1A1LMNAHTTMCOLN3
SCHEMBL4781526 0.84 MEN1 (0.48) PKMALDH1A1LMNAHTTCCR9
SCHEMBL3098055 0.83 AXL (0.52) KMT2AMEN1GAAKEAP1NFE2L2
SCHEMBL4780415 0.82 MEN1 (0.57) ALDH1A1LMNAL3MBTL1KDM4EKMT2A
SCHEMBL4779121 0.82 KEAP1 (0.45) PKMFFAR4ALDH1A1LMNAHTT
SCHEMBL3083474 0.81 DNMT1 (0.46) ALDH1A1LMNAHTTL3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008008374-A2 CCR2 INHIBITORS AND METHODS OF USE THEREOF CHEMOCENTRYX, INC. (US) 2008-01-17 WO claimed
WO-2008008374-A2 CCR2 INHIBITORS AND METHODS OF USE THEREOF CHEMOCENTRYX, INC. (US) 2008-01-17 WO disclosed