SCHEMBL4776345

SCHEMBL4776345

CN(C)C(=O)CN1C[C@H](C(=O)c2ccccc2)C(c2cccc(O)c2)[C@@H](C(=O)c2ccccc2)C1.CN(C)C(=O)CN1C[C@H](C(=O)c2ccccc2)C(c2ccccc2O)[C@@H](C(=O)c2ccccc2)C1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 10/20 0.39
HTR1A P08908 2/20 0.37
DRD1 P21728 2/20 0.37
DRD4 P21917 2/20 0.37
DRD5 P21918 2/20 0.37
DRD3 P35462 2/20 0.37
DRD2 P14416 1/20 0.37
ABL1 P00519 1/20 0.36
EGFR P00533 1/20 0.36
LCK P06239 1/20 0.36
SRC P12931 1/20 0.36
ABL2 P42684 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
GRIN2B Q13224 1/20 0.36
ESRRG P62508 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4776354 1.00 KIF11 (0.39) KIF11HTR1ADRD1DRD4DRD5
SCHEMBL4020120 0.93 GRIN2B (0.40) KIF11HTR1ADRD1DRD4DRD5
SCHEMBL4020117 0.93 GRIN2B (0.40) KIF11HTR1ADRD1DRD4DRD5
SCHEMBL4026439 0.90 TERT (0.40)
SCHEMBL4026443 0.90 TERT (0.40)
SCHEMBL4813149 0.83 KMO (0.42) DRD3DRD2OPRD1GRIN2B
SCHEMBL4024572 0.83 RORC (0.43) DRD4GRIN2B
SCHEMBL4019712 0.83 RORC (0.43) DRD4GRIN2B
SCHEMBL4019710 0.83 RORC (0.43) DRD4GRIN2B
SCHEMBL4024492 0.82 DRD2 (0.43) DRD1DRD4DRD5DRD3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1962846-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-09-03 EP claimed
WO-2007059323-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-24 WO claimed
EP-1962846-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-09-03 EP disclosed
WO-2007059323-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-24 WO disclosed