SCHEMBL4776382

SCHEMBL4776382

c1ccc2nc3[nH]c(-c4c[nH]c5ccccc45)cc3nc2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.56
ALDH1A1 P00352 2/20 0.56
MAPT P10636 2/20 0.56
LMNA P02545 1/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
GPR55 Q9Y2T6 1/20 0.56
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
PDGFRB P09619 2/20 0.49
PDGFRA P16234 1/20 0.49
TUBB4A P04350 1/20 0.45
TUBB P07437 1/20 0.45
TUBA3C P0DPH7 1/20 0.45
TUBA1B P68363 1/20 0.45
TUBA4A P68366 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4725465 0.84 PDGFRB (0.55) SMN1; SMN2ALDH1A1MAPTLMNACYP1A2
SCHEMBL1778743 0.79 GSK3B (0.61) SMN1; SMN2ALDH1A1MAPTLMNACYP1A2
SCHEMBL1748617 0.75 RIPK1 (0.57) PDGFRBPDGFRATDO2ADRA1AADRA1B
SCHEMBL2476987 0.74 CHEK1 (0.54) SMN1; SMN2ALDH1A1MAPTLMNACYP1A2
SCHEMBL4776375 0.73 RAB9A (0.50) SMN1; SMN2ALDH1A1MAPTCYP1A2CYP2C9
SCHEMBL5942610 0.71 CCNB2 (0.58) SMN1; SMN2ALDH1A1MAPTLMNACYP1A2
SCHEMBL8033955 0.70 MEN1 (0.63) SMN1; SMN2ALDH1A1MAPTLMNACYP1A2
SCHEMBL1202543 0.69 IMPDH2 (0.63) SMN1; SMN2ALDH1A1MAPTLMNACYP1A2
SCHEMBL1902587 0.69 MEN1 (1.00) SMN1; SMN2ALDH1A1MAPTLMNACYP1A2
SCHEMBL1748962 0.68 IMPDH2 (0.47) KMT2ATDO2ADRA1AADRA1BHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008014249-A2 IMPROVED PREPARATIONS OF 2 -SUBSTITUTED PYRROLO [2, 3-B] PYRAZINE ( 4, 7 -DIAZAINDOLE ) COMPOUNDS SANOFI-AVENTIS (FR) 2008-01-31 WO disclosed