SCHEMBL4778112

SCHEMBL4778112

CC(C)Cc1nc(CCCc2ccccc2)cc(-c2ccc(N)cc2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.47
NOS1 P29475 1/20 0.47
NOS2 P35228 1/20 0.47
MAOB P27338 4/20 0.42
MAPT P10636 3/20 0.41
MEN1 O00255 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
KMT2A Q03164 2/20 0.41
XDH P47989 1/20 0.38
DHODH Q02127 1/20 0.38
ACHE P22303 1/20 0.38
LTB4R Q15722 1/20 0.38
GSK3B P49841 2/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
GLA P06280 1/20 0.37
MAOA P21397 2/20 0.37
HRH4 Q9H3N8 1/20 0.37
CTSS P25774 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4778391 0.82 NOS3 (0.38) NOS3NOS1NOS2MAPTMEN1
SCHEMBL4774798 0.75 NOS3 (0.42) NOS3NOS1NOS2MAOBMAPT
SCHEMBL4796742 0.75 MAOA (0.47) MAOBMAOA
SCHEMBL22086956 0.73 ADORA1 (0.51) MAPTMEN1ALDH1A1HPGDKMT2A
SCHEMBL4778323 0.72 NOS3 (0.43) NOS3NOS1NOS2MAOBMAPT
SCHEMBL4774672 0.72 NOS3 (0.43) NOS3NOS1NOS2MAOBMAPT
SCHEMBL4774100 0.71 NOS3 (0.42) NOS3NOS1NOS2MAOBMAPT
SCHEMBL4781142 0.71 ALDH1A1 (0.48) NOS3NOS1NOS2MAOBMAPT
SCHEMBL4774626 0.71 NOS3 (0.43) NOS3NOS1NOS2MAOBMAPT
SCHEMBL4776700 0.71 HRH2 (0.42) NOS3NOS1NOS2MAOBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed