SCHEMBL4780097

SCHEMBL4780097

Cc1cccc(C2[C@@H](C(=O)c3ccccc3)CN(CCN(C)C)C[C@@H]2C(=O)c2ccccc2)c1C

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 5/20 0.41
HRH3 Q9Y5N1 2/20 0.40
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
KCNH2 Q12809 1/20 0.35
RORC P51449 1/20 0.35
ACHE P22303 1/20 0.34
P2RX7 Q99572 1/20 0.34
CCR5 P51681 1/20 0.34
SLC6A1 P30531 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4778087 0.94 KIF11 (0.47) KIF11HRH3KCNH2ACHEP2RX7
SCHEMBL4021692 0.89 ALDH1A1 (0.38) KIF11KDM4EALDH1A1
SCHEMBL4780207 0.87 L3MBTL1 (0.37) KIF11ALDH1A1KCNH2RORCCCR5
SCHEMBL4772352 0.87 L3MBTL1 (0.37) KIF11ALDH1A1KCNH2RORCCCR5
SCHEMBL4776377 0.87 KCNH2 (0.42) KIF11ALDH1A1KCNH2RORC
SCHEMBL4026853 0.87 KIF11 (0.38) KIF11HRH3RORC
SCHEMBL4019939 0.87 KIF11 (0.38) KIF11HRH3RORC
SCHEMBL4019937 0.87 KIF11 (0.38) KIF11HRH3RORC
SCHEMBL4024639 0.87 OPRM1 (0.36) KIF11HRH3KCNH2RORCCCR5
SCHEMBL4024642 0.87 OPRM1 (0.36) KIF11HRH3KCNH2RORCCCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1962846-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-09-03 EP claimed
WO-2007059323-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-24 WO claimed