SCHEMBL4780927

SCHEMBL4780927

COc1ccc2ncc(C(=O)C=CC34CC5CC(CC(C5)C3)C4)cc2c1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.46
F2 P00734 1/20 0.46
GLA P06280 1/20 0.46
HPGD P15428 1/20 0.46
HPGDS O60760 13/20 0.44
CYP3A4 P08684 2/20 0.41
EGFR P00533 1/20 0.41
TNFRSF1A P19438 1/20 0.40
CYP1A1 P04798 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP1B1 Q16678 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4731545 1.00 ALDH1A1 (0.46) ALDH1A1F2GLAHPGDHPGDS
SCHEMBL4728653 0.92 HPGDS (0.54) HPGDS
SCHEMBL4729592 0.85 PDGFRB (0.42) ALDH1A1HPGDSEGFR
SCHEMBL5511161 0.82 MGAM (0.49) ALDH1A1HPGDS
SCHEMBL6093635 0.79 CNR2 (0.55) ALDH1A1HPGDTNFRSF1ACYP1B1
SCHEMBL5505975 0.77 MEN1 (0.58) ALDH1A1HPGDCYP3A4CYP1A1CYP1A2
SCHEMBL4730336 0.77 ALDH1A1 (0.36) ALDH1A1HPGDCYP3A4CYP1A1CYP1A2
SCHEMBL4730657 0.77 MAPT (0.35) ALDH1A1HPGD
SCHEMBL5504502 0.76 ABCG2 (0.50) CYP1A1CYP1A2CYP2D6CYP1B1
SCHEMBL4729401 0.76 MAOA (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008035049-A1 ADAMANTANYL-(CYCLOPROPYL)-KETONES AS METABOTROPIC GLUTAMATE RECEPTOR MODULATORS MERZ PHARMA GMBH & CO. KGAA (DE) 2008-03-27 WO disclosed