SCHEMBL4782354

SCHEMBL4782354

Cc1nc2c3c(c(C(=O)N(C)C)cc2n1C)CCC1(Cc2ccccc2C1)O3

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
GLA P06280 1/20 0.31
AKR1C3 P42330 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4739107 0.91 ALDH1A1 (0.31) ALDH1A1
SCHEMBL4738609 0.89 DHODH (0.36) KDM4EALDH1A1KMT2A
SCHEMBL4735029 0.87 NPY5R (0.33) KDM4EALDH1A1
SCHEMBL4739802 0.86 NPC1 (0.32)
SCHEMBL4734384 0.85 KMT2A (0.36) ALDH1A1GLAKMT2A
SCHEMBL4737070 0.85 ALDH1A1 (0.36) KDM4EALDH1A1GLAKMT2A
SCHEMBL14068756 0.84
SCHEMBL4734073 0.84 CHIA (0.33) KDM4E
SCHEMBL13983102 0.83 HRH3 (0.31)
SCHEMBL4737882 0.83 RAB9A (0.35) KDM4EALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071765-A1 PHARMACEUTICALLY ACTIVE SPIRO-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES NYCOMED GMBH (DE) 2008-06-19 WO claimed