SCHEMBL479736

SCHEMBL479736

Cc1cc(C(O)(C(C)c2ccc(OC(C)(C)C(=O)O)c(Cl)c2Cl)C(F)(F)F)c[nH]c1=O

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 2/20 0.35
PPARD Q03181 18/20 0.33
PPARA Q07869 18/20 0.33
PPARG P37231 12/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL479942 0.90 FBP1 (0.38) PTGDR2PPARA
SCHEMBL480100 0.83 PTGER4 (0.35)
SCHEMBL479197 0.81 SCN8A (0.34) PPARDPPARAPPARG
SCHEMBL479998 0.79 ALDH1A1 (0.34)
SCHEMBL479879 0.79 ACACB (0.32)
SCHEMBL733521 0.78 PPARD (0.34) PTGDR2PPARDPPARAPPARG
SCHEMBL753132 0.78 PPARD (0.34) PTGDR2PPARDPPARAPPARG
SCHEMBL479923 0.77 SCN8A (0.36) PPARDPPARAPPARG
SCHEMBL480094 0.76 ACACB (0.32)
SCHEMBL479715 0.74 IGFBP3 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP claimed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO claimed
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed