SCHEMBL479197

SCHEMBL479197

Cc1cc(C(O)(C(C)c2ccc(Oc3ccc(C(=O)O)c(F)c3)c(Cl)c2Cl)C(F)(F)F)c[nH]c1=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN8A Q9UQD0 5/20 0.34
SCN10A Q9Y5Y9 5/20 0.34
PPARG P37231 6/20 0.33
PPARD Q03181 6/20 0.33
PPARA Q07869 6/20 0.33
MEN1 O00255 1/20 0.32
TTR P02766 1/20 0.32
PPOX P50336 1/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
FFAR1 O14842 1/20 0.31
CYP2C9 P11712 1/20 0.31
KCNH2 Q12809 1/20 0.31
CACNA1C Q13936 1/20 0.31
RHEB Q15382 1/20 0.31
PRKAB2 O43741 1/20 0.31
PRKAG1 P54619 1/20 0.31
PRKAA2 P54646 1/20 0.31
PRKAA1 Q13131 1/20 0.31
PRKAG3 Q9UGI9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL479923 0.92 SCN8A (0.36) SCN8ASCN10APPARGPPARDPPARA
SCHEMBL480020 0.90 PRKAB2 (0.33) PPARGPPARDPPARAPRKAB2PRKAG1
SCHEMBL480037 0.89 SCN8A (0.34) SCN8ASCN10APPARGPPARDPPARA
SCHEMBL480100 0.89 PTGER4 (0.35) FFAR1RHEBBRD4
SCHEMBL479915 0.88 PRKAB2 (0.33) PPARGPPARDPPARAMEN1KMT2A
SCHEMBL479998 0.84 ALDH1A1 (0.34) SCN8ASCN10ABRD4
SCHEMBL479931 0.83 S1PR2 (0.33) PPARGPPARDPPARAMEN1TTR
SCHEMBL479715 0.82 IGFBP3 (0.35) FFAR1KCNH2
SCHEMBL480013 0.81 RXRB (0.35) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL733103 0.81 SCN8A (0.35) SCN8ASCN10APPARGPPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP claimed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO claimed
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed