SCHEMBL479739

SCHEMBL479739

COC(=O)c1ccc(Oc2ccc(Cl)c(C(C)C(O)(c3c[nH]c(=O)c(C)c3)C(F)(F)F)c2)cc1Cl

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.33
PDK2 Q15119 1/20 0.31
HTR2A P28223 1/20 0.31
SLC6A4 P31645 1/20 0.31
KCNH2 Q12809 1/20 0.31
KMT2A Q03164 2/20 0.31
ATM Q13315 1/20 0.31
BTK Q06187 1/20 0.31
SCN8A Q9UQD0 1/20 0.31
SCN10A Q9Y5Y9 1/20 0.31
TP53 P04637 1/20 0.30
MAPT P10636 1/20 0.30
MEN1 O00255 1/20 0.30
PKM P14618 1/20 0.30
PPARG P37231 1/20 0.30
PPARD Q03181 1/20 0.30
PPARA Q07869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL479964 0.94 KDR (0.32) KDRPDK2KMT2AATMBTK
SCHEMBL479721 0.93 P2RX3 (0.34) KDRSCN8ASCN10A
SCHEMBL480000 0.91 S1PR2 (0.33) HTR2ASLC6A4KCNH2KMT2ABTK
SCHEMBL480031 0.86 KMT2A (0.32) KMT2AMAPTMEN1PKM
SCHEMBL479915 0.86 PRKAB2 (0.33) KMT2AMEN1PKMPPARGPPARD
SCHEMBL479970 0.86 CYP4F2 (0.37) KMT2AMEN1PKM
SCHEMBL479983 0.85 KDR (0.36) KDRPDK2KMT2AMAPTMEN1
SCHEMBL479931 0.85 S1PR2 (0.33) KMT2ABTKMEN1PPARGPPARD
SCHEMBL480079 0.85 PDK2 (0.40) PDK2MAPT
SCHEMBL479741 0.84 MET (0.36) KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP claimed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO claimed
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed