SCHEMBL479741

SCHEMBL479741

Cc1cc(C(O)(C(C)c2cc(Oc3ccc(F)c(C(=O)O)c3)ccc2Cl)C(F)(F)F)c[nH]c1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 5/20 0.36
ADRA2A P08913 1/20 0.33
CLCN2 P51788 1/20 0.33
ADRB1 P08588 1/20 0.33
ADRB3 P13945 1/20 0.33
P2RX3 P56373 1/20 0.32
MRGPRX4 Q96LA9 1/20 0.32
NTRK1 P04629 1/20 0.32
PRKAB2 O43741 1/20 0.32
PRKAG1 P54619 1/20 0.32
PRKAA2 P54646 1/20 0.32
PRKAA1 Q13131 1/20 0.32
PRKAG3 Q9UGI9 1/20 0.32
PRKAG2 Q9UGJ0 1/20 0.32
PRKAB1 Q9Y478 1/20 0.32
MEN1 O00255 1/20 0.31
TTR P02766 1/20 0.31
PPOX P50336 1/20 0.31
KMT2A Q03164 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL480031 0.94 KMT2A (0.32) METADRB1ADRB3MRGPRX4PRKAB2
SCHEMBL479915 0.93 PRKAB2 (0.33) METADRA2ACLCN2P2RX3NTRK1
SCHEMBL480000 0.91 S1PR2 (0.33) METADRA2ACLCN2PRKAB2PRKAG1
SCHEMBL479871 0.91 MRGPRX4 (0.33) METP2RX3MRGPRX4MEN1KMT2A
SCHEMBL479721 0.86 P2RX3 (0.34) METP2RX3NTRK1
SCHEMBL480020 0.86 PRKAB2 (0.33) METADRA2ACLCN2P2RX3PRKAB2
SCHEMBL479970 0.86 CYP4F2 (0.37) MRGPRX4MEN1KMT2A
SCHEMBL479931 0.85 S1PR2 (0.33) ADRA2ACLCN2PRKAB2PRKAG1PRKAA2
SCHEMBL479739 0.84 KDR (0.33) MEN1KMT2A
SCHEMBL480037 0.84 SCN8A (0.34) METPRKAB2PRKAG1PRKAA2PRKAA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP claimed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO claimed
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed