SCHEMBL479790

SCHEMBL479790

Cc1cc(C(O)(C(C)c2ccc(Oc3ccc(F)c(OCC(=O)O)c3)cc2Cl)C(F)(F)F)c[nH]c1=O

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.36
PPARD Q03181 12/20 0.35
FFAR1 O14842 5/20 0.34
PPARG P37231 3/20 0.34
PPARA Q07869 2/20 0.34
NR3C1 P04150 1/20 0.33
THRA P10827 1/20 0.33
THRB P10828 1/20 0.33
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL479674 0.92 PPOX (0.33) THRATHRBCYP2C19
SCHEMBL479958 0.91 MCL1 (0.41) MCL1PPARDFFAR1PPARGPPARA
SCHEMBL480020 0.84 PRKAB2 (0.33) PPARDPPARGPPARA
SCHEMBL479852 0.84 SMN1; SMN2 (0.40) PPARDFFAR1PPARGPPARATHRA
SCHEMBL480101 0.84 MCL1 (0.35) MCL1FFAR1THRATHRB
SCHEMBL479931 0.83 S1PR2 (0.33) PPARDPPARGPPARATHRATHRB
SCHEMBL732947 0.83 CYP2C19 (0.35) PPARDFFAR1PPARGPPARANR3C1
SCHEMBL753291 0.83 CYP2C19 (0.35) PPARDFFAR1PPARGPPARANR3C1
SCHEMBL479912 0.83 THRB (0.35) THRATHRB
SCHEMBL480172 0.82 NR3C1 (0.34) MCL1PPARDFFAR1PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP claimed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO claimed
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed