SCHEMBL4807472

SCHEMBL4807472

O=C(CC1CCCN(S(=O)(=O)c2ccc(F)cc2)C1)ONNC(=O)c1ccc(Cl)cc1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.50
CYP2C19 P33261 1/20 0.50
KMT2A Q03164 5/20 0.47
MAPT P10636 5/20 0.47
HTT P42858 4/20 0.47
LMNA P02545 3/20 0.47
GAA P10253 1/20 0.47
MEN1 O00255 2/20 0.45
NPY1R P25929 1/20 0.45
NPY2R P49146 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
FLT1 P17948 1/20 0.44
FLT4 P35916 1/20 0.44
KDR P35968 1/20 0.44
TSHR P16473 2/20 0.42
KDM4E B2RXH2 1/20 0.42
HSD17B10 Q99714 1/20 0.42
POLB P06746 3/20 0.42
ALDH1A1 P00352 2/20 0.42
CYP19A1 P11511 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4740406 0.92 ALDH1A1 (0.44) KMT2AHTTLMNAGAAMEN1
SCHEMBL4740126 0.86 CCR1 (0.44) MAPTHTTLMNANPSR1FLT1
SCHEMBL4741276 0.84 TSHR (0.41) KMT2AMAPTHTTLMNANPSR1
SCHEMBL4795192 0.83 CYP3A4 (0.55) CYP3A4CYP2C19KMT2AMAPTHTT
SCHEMBL4739855 0.81 KMT2A (0.58) CYP3A4CYP2C19KMT2AMAPTHTT
SCHEMBL4740909 0.76 CYP2C19 (0.46) CYP2C19KMT2AGAAMEN1HSD17B10
SCHEMBL4740080 0.76 GAA (0.47) CYP2C19MAPTHTTLMNAGAA
SCHEMBL4787140 0.76 POLB (0.51) CYP3A4CYP2C19KMT2ALMNAGAA
SCHEMBL4807466 0.75 CYP3A4 (0.54) CYP3A4CYP2C19KMT2AMAPTHTT
SCHEMBL4741026 0.74 ALDH1A1 (0.52) CYP2C19KMT2ALMNAGAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008087654-A2 PIPERIDINES AS INHIBITORS OF 11β-HYDROXYSTEROID DEHYDROGENASE TYPE 1 CADILA HEALTHCARE LIMITED (IN) 2008-07-24 WO disclosed