SCHEMBL4740126

SCHEMBL4740126

O=C(CC1CCCN(S(=O)(=O)c2ccccc2Cl)C1)ONNC(=O)c1ccc(Cl)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 2/20 0.44
POLB P06746 1/20 0.44
FLT1 P17948 1/20 0.43
FLT4 P35916 1/20 0.43
KDR P35968 1/20 0.43
ATM Q13315 1/20 0.41
FAAH O00519 2/20 0.41
TSHR P16473 1/20 0.41
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4741276 0.93 TSHR (0.41) CCR1POLBFLT1FLT4KDR
SCHEMBL4740406 0.86 ALDH1A1 (0.44) POLBFLT1FLT4KDRHTT
SCHEMBL4807472 0.86 CYP3A4 (0.50) POLBFLT1FLT4KDRTSHR
SCHEMBL4736817 0.82 HTT (0.46) CCR1POLBATMFAAHTSHR
SCHEMBL4740123 0.78 CCR1 (0.47) CCR1POLBATMFAAHTSHR
SCHEMBL4740909 0.75 CYP2C19 (0.46)
SCHEMBL4740080 0.75 GAA (0.47) POLBHTTNPSR1LMNAMAPT
SCHEMBL4736733 0.75 HSD11B1 (0.51) TSHRHTTNPSR1HDAC3HDAC4
SCHEMBL4787140 0.74 POLB (0.51) POLBLMNA
SCHEMBL4738916 0.73 HDAC3 (0.52) CCR1POLBFAAHTSHRHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008087654-A2 PIPERIDINES AS INHIBITORS OF 11β-HYDROXYSTEROID DEHYDROGENASE TYPE 1 CADILA HEALTHCARE LIMITED (IN) 2008-07-24 WO disclosed