SCHEMBL4740909

SCHEMBL4740909

Cc1ccc(C(=O)NNOC(=O)CC2CCCN(S(=O)(=O)c3ccccc3)C2)c(C)c1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.46
HSD17B10 Q99714 1/20 0.44
ALDH1A1 P00352 3/20 0.42
GAA P10253 3/20 0.41
USP2 O75604 2/20 0.40
MAPK1 P28482 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4736655 0.87 HSD17B10 (0.47) CYP2C19HSD17B10ALDH1A1GAAUSP2
SCHEMBL4741026 0.86 ALDH1A1 (0.52) CYP2C19ALDH1A1GAAUSP2MAPK1
SCHEMBL4740080 0.85 GAA (0.47) CYP2C19HSD17B10ALDH1A1GAAUSP2
SCHEMBL4787140 0.84 POLB (0.51) CYP2C19HSD17B10ALDH1A1GAAUSP2
SCHEMBL4740406 0.83 ALDH1A1 (0.44) ALDH1A1GAAUSP2MAPK1MEN1
SCHEMBL4795192 0.79 CYP3A4 (0.55) CYP2C19HSD17B10ALDH1A1GAAMEN1
SCHEMBL4740908 0.78 P2RX7 (0.49) CYP2C19HSD17B10GAAUSP2MAPK1
SCHEMBL4740423 0.77 SIRT2 (0.48) ALDH1A1GAAUSP2MEN1KMT2A
SCHEMBL4807472 0.76 CYP3A4 (0.50) CYP2C19HSD17B10ALDH1A1GAAMEN1
SCHEMBL4740126 0.75 CCR1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008087654-A2 PIPERIDINES AS INHIBITORS OF 11β-HYDROXYSTEROID DEHYDROGENASE TYPE 1 CADILA HEALTHCARE LIMITED (IN) 2008-07-24 WO claimed