Eglumetad

Eglumetad

SCHEMBL481248

N[C@@]1(C(=O)O)CC[C@H]2[C@H](C(=O)O)[C@H]21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 14/20 1.00
GRM3 Q14832 14/20 1.00
GRM6 O15303 11/20 1.00
GRM8 O00222 7/20 1.00
SLC1A2 P43004 1/20 0.73
SLC1A1 P43005 1/20 0.73
GRM4 Q14833 2/20 0.46
GRM1 Q13255 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Eglumetad SCHEMBL13319987 1.00 GRM2 (1.00) GRM2GRM3GRM6GRM8SLC1A2
Eglumetad SCHEMBL15060586 1.00 GRM2 (1.00) GRM2GRM3GRM6GRM8SLC1A2
Eglumetad SCHEMBL16585263 1.00 GRM2 (1.00) GRM2GRM3GRM6GRM8SLC1A2
Eglumetad SCHEMBL13728495 1.00 GRM2 (1.00) GRM2GRM3GRM6GRM8SLC1A2
Eglumetad SCHEMBL231157 1.00 GRM2 (1.00) GRM2GRM3GRM6GRM8SLC1A2
Eglumetad SCHEMBL1650783 0.98 GRM2 (0.96) GRM2GRM3GRM6GRM8SLC1A2
SCHEMBL30417494 0.85 SLC1A2 (1.00) GRM2GRM3GRM6GRM8SLC1A2
SCHEMBL6697973 0.80 GRM2 (0.67) GRM2GRM3GRM6GRM8SLC1A2
Hydrochloric Acid SCHEMBL4810986 0.79 SLC1A2 (0.66) GRM2GRM3GRM6GRM8SLC1A2
Hydrochloric Acid SCHEMBL6699648 0.79 GRM2 (0.65) GRM2GRM3GRM6GRM8SLC1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 88 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023097186-A1 COMPOSITIONS AND METHODS FOR ENHANCING VISUAL FUNCTION THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-06-01 WO claimed
EP-2704793-B1 REGULATION OF AMYLOID BETA MOLECULAR COMPOSITION FOR THE TREATMENT OF ALZHEIMER'S DISEASE UNIV RAMOT (IL) 2019-07-17 EP claimed
US-20250295713-A1 COMPOSITIONS AND METHODS FOR IMPROVING SKIN HEALTH AND FOR THE TREATMENT AND PREVENTION OF DISEASES, DISORDERS AND CONDITIONS ASSOCIATED WITH PATHOGENIC MICROBES DERMBIONT, INC. 2025-09-25 US disclosed
EP-4584250-A1 COMBINATION THERAPIES INCLUDING METAL CHANNEL ACTIVATORS Biohaven Therapeutics Ltd. (VG) 2025-07-16 EP disclosed
US-20250152601-A1 Compositions and Methods for the Treatment of Sexual Dysfunctions THE JONATHAN HURT LIVING TRUST (US) 2025-05-15 US disclosed
US-12064459-B2 Compositions and methods for improving skin health and for the treatment and prevention of diseases, disorders and conditions associated with pathogenic microbes DERMBIONT, INC. (US) 2024-08-20 US disclosed
US-11938106-B2 Treatment of tinnitus using glutamate receptor agonists NORTHEAST OHIO MEDICAL UNIVERSITY (US) 2024-03-26 US disclosed
WO-2024054811-A1 COMBINATION THERAPIES INCLUDING METAL CHANNEL ACTIVATORS BIOHAVEN THERAPEUTICS LTD. (VG) 2024-03-14 WO disclosed
US-20240074995-A1 METHODS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH AN ABNORMAL INFLAMMATORY RESPONSES FIRST WAVE BIO, INC. 2024-03-07 US disclosed
US-11793777-B2 Methods and compositions for treating conditions associated with an abnormal inflammatory response FIRST WAVE BIO, INC. (US) 2023-10-24 US disclosed
US-11744812-B2 Methods of treatment FIRST WAVE BIO, INC. (US) 2023-09-05 US disclosed
EP-1110943-B1 6-FLUOROBICYCLO 3. 1.0]HEXANE DERIVATIVES TAISHO PHARMACEUTICAL CO LTD (JP) 2004-06-16 EP disclosed
US-20040077879-A1 Bis (amino acid) molecular scaffolds UNIVERSITY OF PITTSBURGH - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION 2004-04-22 US disclosed
US-20040006114-A1 Potentiators of glutamate receptors ELI LILLY AND COMPANY 2004-01-08 US disclosed
WO-2003045898-A1 PRODRUGS OF EXCITATORY AMINO ACIDS ELI LILLY AND COMPANY (US) 2003-06-05 WO disclosed
EP-1052246-B1 FLUORINE-CONTAINING AMINO ACID DERIVATIVES TAISHO PHARMACEUTICAL CO LTD (JP) 2003-04-02 EP disclosed
US-6333428-B1 TREATMENT OR PREVENTION OF PSYCHIATRIC DISORDERS OR NEUROLOGICAL DISEASES TAISHO PHARMACEUTICAL CO., LTD. (JP) 2001-12-25 US disclosed
US-6316498-B1 FOR THERAPY AND PROPHYLAXIS OF PSYCHIATRIC DISORDERS SUCH AS SCHIZOPHRENIA, ANXIETY, ASSOCIATED DISEASES, DEPRESSION, BIPOLAR DISTURBANCE AND EPILEPSY, NEUROLOGICAL DISEASES SUCH AS DRUG ADDICTION, COGNITION DISORDER, ALZHEIMER'S DISEASE TAISHO PHARMACEUTICAL CO., LTD. (JP) 2001-11-13 US disclosed
EP-1110943-A1 6-FLUOROBICYCLO 3. 1.0]HEXANE DERIVATIVES Taisho Pharmaceutical Co. Ltd. (JP) 2001-06-27 EP disclosed
EP-1052246-A1 FLUORINE-CONTAINING AMINO ACID DERIVATIVES TAISHO PHARMACEUTICAL CO., LTD (JP) 2000-11-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040077879-A1 Bis (amino acid) molecular scaffolds DNPEP, BCAT1, BCAT2 GRM2 1639/4885GRM3 663/4885GRM6 1882/4885
US-20240074995-A1 METHODS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH AN ABNORMAL INFLAMMATORY RESPONSES FH, CS, ECHS1 GRM2 682/4885GRM3 977/4885GRM6 562/4885
US-11744812-B2 Methods of treatment ACE2, ACE, SI GRM2 130/4885GRM3 125/4885GRM6 583/4885
US-11793777-B2 Methods and compositions for treating conditions associated with an abnormal inflammatory response FH, CS, ECHS1 GRM2 718/4885GRM3 1016/4885GRM6 570/4885
US-20040006114-A1 Potentiators of glutamate receptors GRM1, GRIN1, GRM2 GRM2 3/4885GRM3 6/4885GRM6 13/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.