SCHEMBL4819780

SCHEMBL4819780

[CH2]C(C)CCc1cccc2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.47
CYP2C19 P33261 2/20 0.47
CYP2D6 P10635 1/20 0.47
SIGMAR1 Q99720 2/20 0.47
SLC18A2 Q05940 1/20 0.46
NQO2 P16083 1/20 0.46
CYP2C9 P11712 1/20 0.46
KMT2A Q03164 1/20 0.44
MTNR1A P48039 2/20 0.44
ADA P00813 1/20 0.42
TDP1 Q9NUW8 2/20 0.42
ESR1 P03372 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2845252 0.85 ESR1 (0.50) CYP1A2CYP2C19CYP2D6SIGMAR1SLC18A2
Ammonia Solution, Strong SCHEMBL11816347 0.83 ESR1 (0.49) CYP1A2CYP2C19CYP2D6SIGMAR1SLC18A2
SCHEMBL11816697 0.81 SLC6A2 (0.58) CYP1A2CYP2C19CYP2D6SIGMAR1SLC18A2
SCHEMBL7907492 0.81 NQO2 (0.50) CYP1A2CYP2C19CYP2D6SIGMAR1SLC18A2
SCHEMBL2480671 0.81 KMT2A (0.51) CYP1A2CYP2C19CYP2D6SIGMAR1SLC18A2
SCHEMBL4817621 0.81 CYP1A2 (0.50) CYP1A2CYP2C19CYP2D6SIGMAR1SLC18A2
SCHEMBL5252569 0.80 TDP1 (0.46) CYP1A2CYP2C19CYP2D6SIGMAR1SLC18A2
SCHEMBL9859583 0.79 SIGMAR1 (0.48) CYP1A2CYP2C19CYP2D6SIGMAR1SLC18A2
SCHEMBL6754477 0.79 CYP1A2 (0.44) CYP1A2CYP2C19CYP2D6SIGMAR1SLC18A2
SCHEMBL11808889 0.79 CYP1A2 (0.44) CYP1A2CYP2C19CYP2D6SIGMAR1SLC18A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7358396-B2 Preparation of optically active amines BASF AKTIENGESELLSCHAFT (DE) 2008-04-15 US disclosed
US-20070155971-A1 Chiral diphosphorus compounds and their transition metal complexes Source Global, PBC 2007-07-05 US disclosed
US-7193092-B2 Chiral diphosphorus compounds and their transition metal complexes LANXESS DEUTSCHLAND GMBH (DE) 2007-03-20 US disclosed
US-7078226-B1 Method for producing optically active amines BASF AKTIENGESELLSCHAFT (DE) 2006-07-18 US disclosed
US-20060122429-A1 Preparation of optically active amines DITRICH KLAUS 2006-06-08 US disclosed
EP-1400527-B1 Chiral diphosphorus compounds and transition metal complexes thereof LANXESS DEUTSCHLAND GMBH (DE) 2006-03-22 EP disclosed
EP-1398319-B1 Chiral monophosphorus compounds and transition metal complexes thereof LANXESS DEUTSCHLAND GMBH (DE) 2005-11-09 EP disclosed
CN-1204262-C Method for producing optically active amines BASF AG (DE) 2005-06-01 CN disclosed
US-20050080047-A1 Chiral diphosphorus compounds and their transition metal complexes LANXESS DEUTSCHLAND GMBH (DE) 2005-04-14 US disclosed
CN-1195764-C Transition metal complex, preparation method and use thereof BASF AG (DE) 2005-04-06 CN disclosed
CN-1330074-A Transition metal complex, preparation method and use thereof BASF AG (DE) 2002-01-09 CN disclosed
CN-1072227-C Optically active diphosphine ligands BASF AG (DE) 2001-10-03 CN disclosed
EP-0906324-B1 CARBOHYDRATE DERIVATIVES AND THEIR SOLID-PHASE SYNTHESIS BASF AG (DE) 2001-08-01 EP disclosed
US-6242583-B1 COUPLING CARBOHYDRATE COMPOUNDS IN PRESENCE OF PROMOTER TO A FUNCTIONALIZED SOLID SUPPORT BASF AKTIENGESELLSCHAFT (DE) 2001-06-05 US disclosed
WO-2001038292-A2 METHOD FOR PRODUCING OPTICALLY ACTIVE AMINES BASF AKTIENGESELLSCHAFT (DE) 2001-05-31 WO disclosed
US-5990320-A Optically active diphosphine ligands BASF AKTIENGESELLSCHAFT (DE) 1999-11-23 US disclosed
CN-1219937-A Carbohydrate derivatives and their solid-phase synthesis BASF AG (DE) 1999-06-16 CN disclosed
EP-0906324-A1 CARBOHYDRATE DERIVATIVES AND THEIR SOLID-PHASE SYNTHESIS BASF AKTIENGESELLSCHAFT (DE) 1999-04-07 EP disclosed
CN-1202492-A Optically active diphosphine ligands BASF AG (DE) 1998-12-23 CN disclosed
WO-1997045436-A1 CARBOHYDRATE DERIVATIVES AND THEIR SOLID-PHASE SYNTHESIS BASF AKTIENGESELLSCHAFT (DE) 1997-12-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060122429-A1 Preparation of optically active amines MAOA, MAOB, NAAA CYP1A2 165/4885CYP2C19 269/4885CYP2D6 616/4885
US-20070155971-A1 Chiral diphosphorus compounds and their transition metal complexes CDIPT, DCPS, PIN1 CYP1A2 1320/4885CYP2C19 1457/4885CYP2D6 201/4885
US-20050080047-A1 Chiral diphosphorus compounds and their transition metal complexes CDIPT, DCPS, PIN1 CYP1A2 1320/4885CYP2C19 1457/4885CYP2D6 201/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.