SCHEMBL4820134

SCHEMBL4820134

O=CC(=O)N(c1ccncn1)c1c[nH]c2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.43
RAB9A P51151 4/20 0.43
ALDH1A1 P00352 3/20 0.43
TDP1 Q9NUW8 2/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
MITF O75030 1/20 0.43
LMNA P02545 3/20 0.42
NPSR1 Q6W5P4 2/20 0.42
MAPT P10636 2/20 0.40
HTT P42858 1/20 0.40
IMPDH2 P12268 2/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
GPR84 Q9NQS5 1/20 0.35
CYP2A6 P11509 1/20 0.35
PBRM1 Q86U86 1/20 0.34
ATM Q13315 1/20 0.34
KDM4E B2RXH2 1/20 0.34
CDK4 P11802 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4790366 0.83 ALDH1A1 (0.52) NPC1RAB9AALDH1A1TDP1KMT2A
SCHEMBL13730470 0.71 ALDH1A1 (0.42) NPC1RAB9AALDH1A1TDP1KMT2A
SCHEMBL7334283 0.68 ALDH1A1 (0.62) NPC1RAB9AALDH1A1TDP1KMT2A
SCHEMBL7343483 0.67 ALDH1A1 (0.61) NPC1RAB9AALDH1A1TDP1KMT2A
SCHEMBL3718482 0.63 NPSR1 (0.44) NPC1RAB9AALDH1A1TDP1KMT2A
SCHEMBL4592999 0.63 P2RX7 (0.40) ALDH1A1TDP1KMT2AMEN1NPSR1
SCHEMBL6394938 0.63 ALDH1A1 (0.56) NPC1RAB9AALDH1A1TDP1KMT2A
SCHEMBL30378846 0.62 HSD17B10 (0.60) NPC1RAB9AALDH1A1KMT2AMEN1
SCHEMBL9828569 0.62 HSD17B10 (0.60) NPC1RAB9AALDH1A1KMT2AMEN1
3-Formylindole SCHEMBL29082887 0.62 CYP2A6 (0.77) NPC1RAB9AALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008157740-A2 FAAH INHIBITORS IRONWOOD PHARMACEUTICALS, INC. (US) 2008-12-24 WO disclosed