SCHEMBL4820547

SCHEMBL4820547

O=C(NC1Cc2ccccc2CC1O)OCc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
GAA P10253 1/20 0.52
CPB1 P15086 2/20 0.51
TSHR P16473 1/20 0.50
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
ACHE P22303 2/20 0.49
EPHX1 P07099 1/20 0.47
CTSL P07711 1/20 0.45
CTSB P07858 1/20 0.45
CTSK P43235 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14193328 1.00 ALDH1A1 (0.52) ALDH1A1GAACPB1TSHRCA1
SCHEMBL1718206 0.90 CA1 (0.54) ALDH1A1GAACPB1TSHRCA1
SCHEMBL4574080 0.84 CPB1 (0.60) ALDH1A1GAACPB1TSHREPHX1
SCHEMBL4088176 0.82 CPB1 (0.59) ALDH1A1GAACPB1TSHREPHX1
SCHEMBL4088179 0.82 CPB1 (0.59) ALDH1A1GAACPB1TSHREPHX1
SCHEMBL13370746 0.82 CPB1 (0.59) ALDH1A1GAACPB1TSHREPHX1
SCHEMBL4093654 0.82 CPB1 (0.59) ALDH1A1GAACPB1TSHREPHX1
SCHEMBL170233 0.82 ALDH1A1 (0.65) ALDH1A1GAACPB1TSHRCA1
SCHEMBL24324120 0.81 CPB1 (0.61) ALDH1A1GAACPB1TSHREPHX1
SCHEMBL8092161 0.81 ALDH1A1 (0.50) ALDH1A1GAATSHRCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365061-B2 2-Amino-3-functionalized tetralin derivatives and related glycogen phosphorylase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2008-04-29 US disclosed
WO-2006055463-A2 2-AMINO-3-FUNCTIONALIZED TETRALIN DERIVATIVES AND RELATED GLYCOGEN PHOSPHORYLASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2006-05-26 WO disclosed
US-20060111413-A1 Antidiabetic agents, anticancer, non-cardiac ischemia, infection, hypertension, obesity and dislipidemia; 3-(5-chloroindole-2-carbonylamino)-2-hydroxy-1,2,3,4-tetrahydronaphthalene BRISTOL-MYERS SQUIBB COMPANY 2006-05-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060111413-A1 Antidiabetic agents, anticancer, non-cardiac ischemia, infection, hypertension, obesity and dislipidemia; 3-(5-chloroindole-2-carbonylamino)-2-hydroxy-1,2,3,4-tetrahydronaphthalene PYGM, PON1, GYS1 ALDH1A1 1037/4885GAA 872/4885CPB1 581/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.