SCHEMBL4831484

SCHEMBL4831484

CC[N+](C)(CC)C1Cc2cc(Cl)cc(-c3cccc(C)c3C)c2O1

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AQP1 P29972 3/20 0.34
SIRT2 Q8IXJ6 5/20 0.33
EZH2 Q15910 1/20 0.32
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596995 0.79 HTR1A (0.39) AQP1HTR2AHTR2C
SCHEMBL4234706 0.79 AQP1 (0.51) AQP1SIRT2EZH2HTR2AHTR2C
SCHEMBL4596991 0.78 HTR2A (0.37) AQP1SIRT2EZH2HTR2AHTR2C
SCHEMBL4793916 0.77 AQP1 (0.46) AQP1SIRT2EZH2HTR2AHTR2C
SCHEMBL4230246 0.77 AQP1 (0.41) AQP1SIRT2EZH2HTR2AHTR2C
SCHEMBL4230242 0.77 AQP1 (0.58) AQP1SIRT2EZH2HTR2AHTR2C
SCHEMBL4836377 0.76 AQP1 (0.36) AQP1
SCHEMBL4970746 0.74 AQP1 (0.46) AQP1EZH2
SCHEMBL4967601 0.74 AQP1 (0.47) AQP1
SCHEMBL4823949 0.73 AQP1 (0.31) AQP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1871355-A1 NEW THERAPEUTIC COMBIANATIONS FOR THE TREATMENT OR PREVENTION OF DEPRESSION Wyeth (US) 2008-01-02 EP disclosed
WO-2006116149-A1 NEW THERAPEUTIC COMBIANATIONS FOR THE TREATMENT OR PREVENTION OF DEPRESSION WYETH (US) 2006-11-02 WO disclosed