SCHEMBL4970746

SCHEMBL4970746

CC[N+](C)(CC)C1Cc2cc(C)cc(-c3ccc(Cl)cc3Cl)c2O1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AQP1 P29972 2/20 0.46
ALOX15 P16050 2/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
MAPK1 P28482 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CRHR1 P34998 3/20 0.33
F2RL3 Q96RI0 2/20 0.32
HSD11B1 P28845 1/20 0.31
USP2 O75604 1/20 0.30
HSD17B10 Q99714 1/20 0.30
EZH2 Q15910 1/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4836377 0.91 AQP1 (0.36) AQP1ALDH1A1MAPK1USP2KDM4E
SCHEMBL4823949 0.86 AQP1 (0.31) AQP1
SCHEMBL4623489 0.79 AQP1 (0.49) AQP1NPC1ALDH1A1HPGDMAPK1
SCHEMBL4830774 0.78 AQP1 (0.50) AQP1MAPK1
SCHEMBL4623485 0.78 AQP1 (0.48) AQP1NPC1ALDH1A1HPGDCRHR1
SCHEMBL4224721 0.77 AQP1 (0.74) AQP1CRHR1F2RL3HSD11B1EZH2
SCHEMBL4790525 0.76 AQP1 (0.56) AQP1ALOX15NPC1ALDH1A1HPGD
SCHEMBL5605411 0.76 AQP1 (0.46) AQP1NPC1ALDH1A1HPGDMAPK1
SCHEMBL4225189 0.75 AQP1 (0.77) AQP1ALOX15NPC1ALDH1A1HPGD
SCHEMBL5148555 0.75 DRD2 (0.37) ALDH1A1MAPK1F2RL3HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879569-A2 THERAPEUTIC COMBINATIONS FOR THE TREATMENT OR PREVENTION OF PSYCHOTIC DISORDERS Wyeth (US) 2008-01-23 EP disclosed
WO-2006116221-A2 THERAPEUTIC COMBINATIONS FOR THE TREATMENT OR PREVENTION OF PSYCHOTIC DISORDERS WYETH (US) 2006-11-02 WO disclosed