SCHEMBL4836377

SCHEMBL4836377

CC[N+](C)(CC)C1Cc2cc(C)cc(-c3cc(Cl)ccc3Cl)c2O1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AQP1 P29972 2/20 0.36
S1PR4 O95977 2/20 0.31
MAPK1 P28482 2/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
RECQL P46063 1/20 0.31
NPSR1 Q6W5P4 2/20 0.31
MAPT P10636 2/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
USP2 O75604 1/20 0.30
ESR1 P03372 1/20 0.30
HTT P42858 1/20 0.30
GPR55 Q9Y2T6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4970746 0.91 AQP1 (0.46) AQP1MAPK1KDM4EALDH1A1USP2
SCHEMBL4830774 0.87 AQP1 (0.50) AQP1MAPK1NPSR1MAPTTDP1
SCHEMBL4823949 0.86 AQP1 (0.31) AQP1MAPTTDP1
SCHEMBL4766477 0.79 AQP1 (0.39) AQP1S1PR4MAPK1KDM4EALDH1A1
SCHEMBL4766472 0.78 AQP1 (0.38) AQP1S1PR4MAPK1KDM4EALDH1A1
SCHEMBL5140412 0.78 AQP1 (0.37) AQP1S1PR4
SCHEMBL4220746 0.77 AQP1 (0.60) AQP1S1PR4KDM4EALDH1A1MAPT
SCHEMBL4789302 0.76 AQP1 (0.45) AQP1S1PR4
SCHEMBL4831484 0.76 AQP1 (0.34) AQP1
SCHEMBL5606024 0.76 AQP1 (0.37) AQP1S1PR4MAPK1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1871355-A1 NEW THERAPEUTIC COMBIANATIONS FOR THE TREATMENT OR PREVENTION OF DEPRESSION Wyeth (US) 2008-01-02 EP claimed
WO-2006116149-A1 NEW THERAPEUTIC COMBIANATIONS FOR THE TREATMENT OR PREVENTION OF DEPRESSION WYETH (US) 2006-11-02 WO claimed
EP-1871354-A1 TREATMENT OF PAIN Wyeth (US) 2008-01-02 EP disclosed
WO-2006116171-A1 TREATMENT OF PAIN WYETH (US) 2006-11-02 WO disclosed