SCHEMBL4842699

SCHEMBL4842699

COc1c(Cl)ccc(P)c1-c1c(P)ccc(Cl)c1OC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 3/20 0.45
HSD17B10 Q99714 1/20 0.45
TSHR P16473 1/20 0.37
HTR2C P28335 2/20 0.36
HTR2A P28223 1/20 0.36
HTR2B P41595 1/20 0.36
HTR1A P08908 1/20 0.34
HTR1D P28221 1/20 0.34
HTR7 P34969 1/20 0.34
HTR5A P47898 1/20 0.34
TAS1R3 Q7RTX0 5/20 0.33
TAS1R1 Q7RTX1 5/20 0.33
MAPK1 P28482 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
TAS1R2 Q8TE23 3/20 0.33
TUBB4A P04350 1/20 0.33
TUBB P07437 1/20 0.33
TUBA3C P0DPH7 1/20 0.33
TUBA1B P68363 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4657348 0.74 ALDH1A1 (0.48) ALDH1A1KDM4EHSD17B10TSHRHTR2C
SCHEMBL2355429 0.72 ALDH1A1 (0.50) ALDH1A1KDM4EHSD17B10TSHRHTR2C
SCHEMBL29536407 0.72 ALDH1A1 (0.50) ALDH1A1KDM4EHSD17B10TSHRHTR2C
SCHEMBL11484541 0.70 ALDH1A1 (0.48) ALDH1A1KDM4EHSD17B10TSHRHTR2C
SCHEMBL7904037 0.70 AHR (0.42) ALDH1A1KDM4EHSD17B10TSHRHTR2C
SCHEMBL254822 0.69 KDM4E (0.46) ALDH1A1KDM4EHSD17B10TSHRMAPK1
SCHEMBL4657344 0.69 EPHB4 (0.40) ALDH1A1KDM4EHSD17B10TSHRHTR2C
SCHEMBL7713840 0.69 ALDH1A1 (0.43) ALDH1A1KDM4EHSD17B10TSHRHTR2C
SCHEMBL13843510 0.69 CYP2A6 (0.48) ALDH1A1KDM4EHSD17B10TSHRMAPK1
SCHEMBL10945599 0.68 ALDH1A1 (0.47) ALDH1A1KDM4EHSD17B10TSHRHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1636243-B1 CHIRAL LIGANDS FOR APPLICATION IN ASYMMETRIC SYNTHESES BOEHRINGER INGELHEIM INT (DE) 2013-11-06 EP disclosed
US-7396947-B2 Chiral ligands for application in asymmetric syntheses LANXESS DEUTSCHLAND GMBH (DE) 2008-07-08 US disclosed
US-20070004927-A1 Chiral ligands for application in asymmetric syntheses BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-01-04 US disclosed
US-20060161022-A1 Chiral ligands for application in asymmetric syntheses LANXESS DEUTSCHLAND GMBH (DE) 2006-07-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070004927-A1 Chiral ligands for application in asymmetric syntheses COASY, SPR, DHPS ALDH1A1 348/4885KDM4E 4280/4885HSD17B10 178/4885
US-20060161022-A1 Chiral ligands for application in asymmetric syntheses COASY, SPR, DHPS ALDH1A1 348/4885KDM4E 4280/4885HSD17B10 178/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.