SCHEMBL4853514

SCHEMBL4853514

Cc1cc(C)cc(-c2ccc(OCCN(C)C)c(C=CC(=O)c3cccc(O)c3)c2)c1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.47
KDR P35968 4/20 0.46
DPP4 P27487 1/20 0.46
BCHE P06276 4/20 0.44
CHRNA7 P36544 2/20 0.44
ABCG2 Q9UNQ0 1/20 0.42
ACHE P22303 1/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41
P4HB P07237 2/20 0.40
CAPN1 P07384 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4853736 0.90 BCHE (0.52) BCHEACHE
SCHEMBL4856637 0.89 LMNA (0.45) KDRBCHEACHE
SCHEMBL4853345 0.89 RELA (0.48) KDRBCHEACHE
SCHEMBL4852218 0.89 CAPN1 (0.50) DPP4BCHECHRNA7ACHECAPN1
SCHEMBL4846169 0.89 BCHE (0.42) KDRBCHEACHE
SCHEMBL4852888 0.86 HCRTR2 (0.42) KDRBCHEACHE
SCHEMBL4846042 0.86 MAPT (0.50) KDRBCHEACHE
SCHEMBL4846060 0.86 MAPT (0.50) KDRBCHEACHE
SCHEMBL14280884 0.85 BCHE (0.46) BCHEABCG2ACHECAPN1
SCHEMBL4849986 0.85 BCHE (0.46) BCHEABCG2ACHECAPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US claimed
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed