SCHEMBL4855293

SCHEMBL4855293

Cc1cc(N(C)C)ccc1C(c1ccccc1)c1ccc(N(C)C)cc1C.Cc1ccc(N(c2ccc(C)cc2)c2ccc(C=Cc3ccc(C=Cc4ccc(N(c5ccc(C)cc5)c5ccc(C)cc5)cc4)cc3)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RELA Q04206 1/20 0.45
INSR P06213 3/20 0.37
APP P05067 8/20 0.36
MEN1 O00255 3/20 0.36
RAB9A P51151 3/20 0.36
KMT2A Q03164 3/20 0.36
APOBEC3A P31941 2/20 0.36
APOBEC3G Q9HC16 2/20 0.36
NPC1 O15118 2/20 0.36
GAA P10253 1/20 0.36
GFER P55789 1/20 0.36
PTGS1 P23219 1/20 0.35
MAPT P10636 2/20 0.35
TRPM8 Q7Z2W7 2/20 0.35
ALDH1A1 P00352 1/20 0.34
STAT3 P40763 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4855277 1.00 RELA (0.45) RELAINSRAPPMEN1RAB9A
SCHEMBL376187 0.92 ALDH1A1 (0.40) MEN1KMT2AGAAMAPTALDH1A1
SCHEMBL75642 0.84 MAPT (0.41) RELAMEN1RAB9AKMT2ANPC1
SCHEMBL4314898 0.83 MAPT (0.36) MEN1RAB9AKMT2ANPC1GAA
SCHEMBL19886263 0.78 MAPT (0.44) MEN1RAB9AKMT2ANPC1GAA
SCHEMBL13308457 0.76 NFE2L2 (0.45) RELAAPPTRPM8
SCHEMBL12576205 0.76 TRPM8 (0.42) RELAAPPRAB9ANPC1MAPT
SCHEMBL30327005 0.75 MAPT (0.41) MEN1RAB9AKMT2ANPC1GAA
SCHEMBL12120252 0.74 NFE2L2 (0.45) RELAAPPMEN1RAB9AKMT2A
SCHEMBL5921994 0.74 SLC2A1 (0.47) APPKMT2AGAAMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1961055-A2 ELECTROLUMINESCENT DEVICE CONTAINING AN ANTHRACENE DERIVATIVE EASTMAN KODAK COMPANY (US) 2008-08-27 EP disclosed
EP-1941562-A1 ORGANIC ELEMENT FOR LOW VOLTAGE ELECTROLUMINESCENT DEVICES EASTMAN KODAK COMPANY (US) 2008-07-09 EP disclosed
EP-1941563-A2 ORGANIC ELEMENT FOR LOW VOLTAGE ELECTROLUMINESCENT DEVICES EASTMAN KODAK COMPANY (US) 2008-07-09 EP disclosed
EP-1929533-A1 PATTERNING OLED DEVICE ELECTRODES AND OPTICAL MATERIAL EASTMAN KODAK COMPANY (US) 2008-06-11 EP disclosed
EP-1891692-A2 ORGANIC ELEMENT FOR LOW VOLTAGE ELECTROLUMINESCENT DEVICES EASTMAN KODAK COMPANY (US) 2008-02-27 EP disclosed
EP-1833944-A1 ORGANIC ELEMENT FOR ELECTROLUMINESCENT DEVICES EASTMAN KODAK COMPANY (US) 2007-09-19 EP disclosed
WO-2007070251-A2 ELECTROLUMINESCENT DEVICE CONTAINING AN ANTHRACENE DERIVATIVE EASTMAN KODAK COMPANY (US) 2007-06-21 WO disclosed
WO-2007050301-A2 ORGANIC ELEMENT FOR LOW VOLTAGE ELECTROLUMINESCENT DEVICES EASTMAN KODAK COMPANY (US) 2007-05-03 WO disclosed
WO-2007050334-A1 ORGANIC ELEMENT FOR LOW VOLTAGE ELECTROLUMINESCENT DEVICES EASTMAN KODAK COMPANY (US) 2007-05-03 WO disclosed
EP-1779446-A1 DESSICANT FOR TOP-EMITTING OLED EASTMAN KODAK COMPANY (US) 2007-05-02 EP disclosed
WO-2007041116-A1 PATTERNING OLED DEVICE ELECTRODES AND OPTICAL MATERIAL EASTMAN KODAK COMPANY (US) 2007-04-12 WO disclosed
WO-2007005227-A1 ELECTROLUMINESCENT DEVICES CONTAINING BENZIDINE DERIVATIVES EASTMAN KODAK COMPANY (US) 2007-01-11 WO disclosed
WO-2006138075-A2 ORGANIC ELEMENT FOR LOW VOLTAGE ELECTROLUMINESCENT DEVICES EASTMAN KODAK COMPANY (US) 2006-12-28 WO disclosed
WO-2006130353-A2 LIGHT-EMITTING DEVICE CONTAINING BIS-PHOSPHINEOXIDE COMPOUND EASTMAN KODAK COMPANY (US) 2006-12-07 WO disclosed
WO-2006130793-A1 PROCESS FOR MAKING AN ORGANIC LIGHT-EMITTING DEVICE EASTMAN KODAK COMPANY (US) 2006-12-07 WO disclosed
WO-2006033831-A1 ORGANIC ELEMENT FOR ELECTROLUMINESCENT DEVICES EASTMAN KODAK COMPANY (US) 2006-03-30 WO disclosed
WO-2006019857-A1 DESSICANT FOR TOP-EMITTING OLED EASTMAN KODAK COMPANY (US) 2006-02-23 WO disclosed
WO-2005057678-A1 ORGANIC ELECTROLUMINESCENT DEVICES WITH ADDITIVE EASTMAN KODAK COMPANY (US) 2005-06-23 WO disclosed
WO-2005057680-A1 ORGANIC ELEMENT FOR ELECTROLUMINESCENT DEVICES EASTMAN KODAK COMPANY (US) 2005-06-23 WO disclosed
WO-2005020283-A2 WHITE LIGHT-EMITTING DEVICE WITH IMPROVED DOPING EASTMAN KODAK COMPANY (US) 2005-03-03 WO disclosed