SCHEMBL485752

SCHEMBL485752

O=C(NC1CCC1)c1cc(Cl)c2ccccc2c1OCc1csc(-c2cccs2)n1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 14/20 0.46
NPC1 O15118 7/20 0.46
RAB9A P51151 7/20 0.46
PKM P14618 1/20 0.43
SLC6A4 P31645 1/20 0.42
LMNA P02545 2/20 0.41
KMT2A Q03164 3/20 0.40
ALDH1A1 P00352 3/20 0.40
MEN1 O00255 2/20 0.40
MAPT P10636 2/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
TP53 P04637 1/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PBK Q96KB5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL485671 0.88 KDM4E (0.48) KDM4ENPC1RAB9APKMLMNA
Formic Acid SCHEMBL27713042 0.86 SCN9A (0.43) KDM4ERAB9ALMNAKMT2AALDH1A1
SCHEMBL485566 0.83 SHMT1 (0.43) KDM4ENPC1RAB9APKMSLC6A4
SCHEMBL485707 0.77 ALOX5AP (0.51) KDM4ERAB9ALMNAKMT2AALDH1A1
Formic Acid SCHEMBL27713056 0.77 ALOX5AP (0.48) KDM4ERAB9ALMNAKMT2AALDH1A1
SCHEMBL486100 0.76 RAB9A (0.44) KDM4ENPC1RAB9APKMLMNA
SCHEMBL485800 0.76 KMT2A (0.49) KDM4ENPC1RAB9ALMNAKMT2A
Formic Acid SCHEMBL27712967 0.75 KMT2A (0.55) KMT2AALDH1A1MEN1GAA
Formic Acid SCHEMBL27713038 0.75 PIN1 (0.42) KDM4ENPC1RAB9APKMLMNA
SCHEMBL486088 0.74 MRGPRX4 (0.56) KMT2AALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1836158-B1 FUSED BICYCLIC CARBOXAMIDE DERIVATIVES FOR USE AS CXCR2 INHIBITORS IN THE TREATMENT OF INFLAMMATION SANOFI AVENTIS DEUTSCHLAND (DE) 2012-02-01 EP claimed