SCHEMBL4862887

SCHEMBL4862887

O=C(C=NO)c1ccc(Br)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.50
CES1 P23141 1/20 0.50
RAB9A P51151 3/20 0.48
LMNA P02545 2/20 0.48
RECQL P46063 1/20 0.48
MAPT P10636 3/20 0.47
ALDH1A1 P00352 2/20 0.47
CYP1B1 Q16678 1/20 0.47
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
ESR1 P03372 1/20 0.46
ESR2 Q92731 1/20 0.46
GSK3B P49841 2/20 0.43
HTT P42858 1/20 0.43
CYP1A2 P05177 1/20 0.42
NPC1 O15118 2/20 0.42
OGG1 O15527 1/20 0.42
MEN1 O00255 1/20 0.41
STAT1 P42224 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11489877 1.00 CES2 (0.50) CES2CES1RAB9ALMNARECQL
SCHEMBL4862884 1.00 CES2 (0.50) CES2CES1RAB9ALMNARECQL
SCHEMBL28863719 0.83 KMT2A (0.36) RAB9ALMNARECQLMAPTALDH1A1
SCHEMBL9056522 0.80 ALDH5A1 (0.56) CES2RAB9ALMNAMAPTALDH1A1
SCHEMBL4452292 0.80 ALDH5A1 (0.56) CES2RAB9ALMNAMAPTALDH1A1
SCHEMBL1193448 0.78 MEN1 (0.53) CES2CES1RAB9AMAPTCYP1B1
SCHEMBL14842658 0.78 TPMT (0.48) LMNAALDH1A1CA1CA2GSK3B
SCHEMBL12997454 0.78 MEN1 (0.53) CES2CES1RAB9AMAPTCYP1B1
SCHEMBL14842660 0.78 TPMT (0.48) LMNAALDH1A1CA1CA2GSK3B
SCHEMBL11436643 0.78 ALDH1A1 (0.61) CES2CES1RAB9ALMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7470713-B2 Imidazole based kinase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2008-12-30 US disclosed
EP-1175410-B1 PESTICIDAL TRIAZINE DERIVATIVES NOVARTIS AG (CH) 2005-12-07 EP disclosed
US-20050187218-A1 Imidazole based kinase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2005-08-25 US disclosed
US-6723720-B2 PHENYL-SUBSTITUTED 1,2,4-TRIAZINES, ESPECIALLY FOR CONTROLLING FLEAS NOVARTIS ANIMAL HEALTH US, INC. 2004-04-20 US disclosed
US-20030036544-A1 Pesticidal triazine-derivatives NOVARTIS ANIMAL HEALTH US, INC. 2003-02-20 US disclosed
EP-1175410-A1 PESTICIDAL TRIAZINE DERIVATIVES Syngenta Participations AG (CH) 2002-01-30 EP disclosed
WO-2000066568-A1 PESTICIDAL TRIAZINE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2000-11-09 WO disclosed
US-4293552-A Novel 1-(mono-o-substituted benzoyl)-3-(substituted pyrazinyl) ureas ELI LILLY AND COMPANY (US) 1981-10-06 US disclosed
US-4229579-A OPTICAL BRIGHTENERS BAYER AKTIENGESELLSCHAFT (DE) 1980-10-21 US disclosed
US-4160834-A INSECTICIDES ELI LILLY AND COMPANY (US) 1979-07-10 US disclosed
US-4144243-A OPTICAL BRIGHTENERS FOR TEXTILES AND LACQUEARS BAYER AKTIENGESELLSCHAFT (DE) 1979-03-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050187218-A1 Imidazole based kinase inhibitors MAP3K19, MAP3K1, ABL1 CES2 4498/4885CES1 3373/4885RAB9A 1837/4885
US-20030036544-A1 Pesticidal triazine-derivatives DDT, CYCS, TUBA3C CES2 201/4885CES1 194/4885RAB9A 2869/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.