SCHEMBL4865573

SCHEMBL4865573

O=C1CCC(Cc2ccccc2)C1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.48
CYP19A1 P11511 1/20 0.47
SIGMAR1 Q99720 2/20 0.45
HTR1A P08908 1/20 0.45
DDB1 Q16531 1/20 0.45
CRBN Q96SW2 1/20 0.45
NOS3 P29474 1/20 0.45
NOS1 P29475 1/20 0.45
NOS2 P35228 1/20 0.45
CCR3 P51677 2/20 0.44
GRIN2B Q13224 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4865561 1.00 GBA1 (0.48) GBA1CYP19A1SIGMAR1HTR1ADDB1
SCHEMBL3982415 0.89 NOS3 (0.50) GBA1CYP19A1SIGMAR1DDB1CRBN
SCHEMBL5675291 0.88 GBA1 (0.57) GBA1SIGMAR1HTR1ADDB1CRBN
SCHEMBL25698026 0.87 NOS3 (0.45) GBA1CYP19A1SIGMAR1DDB1CRBN
Hydrochloric Acid SCHEMBL28729781 0.84 SIGMAR1 (0.48) GBA1SIGMAR1NOS3NOS1NOS2
SCHEMBL428508 0.84 GBA1 (0.50) GBA1CYP19A1SIGMAR1CCR3GRIN2B
SCHEMBL6517320 0.83 CTSS (0.44)
Bicarbonate SCHEMBL2854194 0.83 GBA1 (0.52) GBA1CCR3
SCHEMBL3699320 0.81 GBA1 (0.50) GBA1SIGMAR1HTR1ADDB1CRBN
SCHEMBL27487290 0.81 ALDH1A1 (0.44) CYP19A1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-218689407-U 2- [4- (2-chloropropionyl) benzyl ] cyclopentanone production device 无棣融川医药化工科技有限公司 2023-03-24 CN disclosed
CN-101168530-B 1,4-dioxoquinoxaline formaldehyde dihydrazone with weed control activity and its preparation method and application UNIV HUAZHONG AGRICULTURAL 2011-02-09 CN disclosed
US-20080125310-A1 Hydride reduction of alpha, beta-unsaturated carbonyl compounds using chiral organic catalysts CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2008-05-29 US disclosed
CN-101168530-A 1,4-dioxoquinoxaline formaldehyde dihydrazone with weed control activity and its preparation method and application UNIV HUAZHONG AGRICULTURAL (CN) 2008-04-30 CN disclosed
US-7323604-B2 Hydride reduction of α,β-unsaturated carbonyl compounds using chiral organic catalysts CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2008-01-29 US disclosed
US-20060161024-A1 Hydride reduction of alpha, beta-unsaturated carbonyl compounds using chiral organic catalysts CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2006-07-20 US disclosed
US-20050065349-A1 Asymmetric 1,4-reductions of and 1,4-additions to enoates and related systems BUCHWALD STEPHEN L (US) 2005-03-24 US disclosed
US-6787655-B2 TRANSITION-METAL-CATALYZED ASYMMETRIC 1,4-ADDITION OF A NUCLEOPHILE, E.G., HYDRIDE, TO CYCLIC AND ACYCLIC ENOATES AND ENONES AND THE CATALYST CONTAINING A COPPER AND AN ASYMMETRIC BIDENTATE BISPHOSPHINE LIGAND MASSACHUSETTS INSTITUTE OF TECHNOLOGY 2004-09-07 US disclosed
US-20030125563-A1 Asymmetric 1,4-reductions of and 1,4-additions to enoates and related systems NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2003-07-03 US disclosed
US-6465664-B1 CATALYZED WITH A TRANSITION METAL CATALYST COMPOSED OF A COPPER COMPOUND AND AN ASYMMETRIC LIGAND, SUCH AS A PHOSPHINE, A NUCLEOPHILE AND A BASE MASSACHUSETTS INSTITUTE OF TECHNOLOGY 2002-10-15 US disclosed
WO-2001019761-A2 ASYMMETRIC 1,4-REDUCTIONS OF AND 1,4-ADDITIONS TO ENOATES AND RELATED SYSTEMS MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2001-03-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050065349-A1 Asymmetric 1,4-reductions of and 1,4-additions to enoates and related systems APEX1, AP2A1, ENPP1 GBA1 1330/4885CYP19A1 93/4885SIGMAR1 3891/4885
US-20030125563-A1 Asymmetric 1,4-reductions of and 1,4-additions to enoates and related systems APEX1, AP2A1, ENPP1 GBA1 1330/4885CYP19A1 93/4885SIGMAR1 3891/4885
US-20060161024-A1 Hydride reduction of alpha, beta-unsaturated carbonyl compounds using chiral organic catalysts ECH1, CBR1, DHCR24 GBA1 945/4885CYP19A1 626/4885SIGMAR1 256/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.