SCHEMBL4866324

SCHEMBL4866324

COc1c(N2CCCC2)cccc1[N+](=O)[O-]

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.50
MAPT P10636 5/20 0.50
CYP1A2 P05177 3/20 0.50
CYP2C19 P33261 3/20 0.50
LMNA P02545 3/20 0.50
GAA P10253 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
HTT P42858 2/20 0.50
CYP3A4 P08684 1/20 0.50
MITF O75030 1/20 0.50
CTSB P07858 1/20 0.50
AR P10275 1/20 0.50
L3MBTL1 Q9Y468 4/20 0.48
KMT2A Q03164 2/20 0.47
NPSR1 Q6W5P4 2/20 0.47
TDP1 Q9NUW8 2/20 0.47
MAPK1 P28482 3/20 0.47
CYP2C9 P11712 1/20 0.47
POLB P06746 1/20 0.47
KDM4E B2RXH2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3643443 0.98 CYP1A2 (0.52) ALDH1A1MAPTCYP1A2CYP2C19LMNA
SCHEMBL8692030 0.88 SIRT6 (0.52) ALDH1A1MAPTCYP1A2CYP2C19LMNA
SCHEMBL24130664 0.87 HTR3A (0.50) ALDH1A1MAPTCYP2C19LMNAGAA
SCHEMBL3722707 0.87 CTSB (0.53) ALDH1A1MAPTCYP1A2CYP2C19LMNA
Hydrochloric Acid SCHEMBL30481714 0.86 MAPT (0.51) ALDH1A1MAPTCYP2C19LMNAGAA
SCHEMBL24130778 0.81 HTT (0.53) ALDH1A1MAPTCYP1A2CYP2C19LMNA
SCHEMBL24133175 0.80 KMT2A (0.41) ALDH1A1MAPTCYP1A2CYP2C19LMNA
SCHEMBL24130446 0.80 MAPT (0.57) ALDH1A1MAPTCYP1A2CYP2C19LMNA
SCHEMBL30481715 0.80 MAPT (0.57) ALDH1A1MAPTCYP1A2CYP2C19LMNA
SCHEMBL3799173 0.79 CTSB (0.65) ALDH1A1MAPTCYP1A2CYP2C19LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1987039-A2 MELANIN CONCENTRATING HORMONE RECEPTOR-1 ANTAGONISTS Brystol-Myers Squibb Company (US) 2008-11-05 EP disclosed
WO-2007092416-A2 MELANIN CONCENTRATING HORMONE RECEPTOR-1 ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-08-16 WO disclosed