SCHEMBL3722707

SCHEMBL3722707

COc1c(N2CCOCC2)cccc1[N+](=O)[O-]

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSB P07858 1/20 0.53
HTT P42858 2/20 0.53
MAPT P10636 9/20 0.51
ALDH1A1 P00352 6/20 0.50
CYP1A2 P05177 3/20 0.50
LMNA P02545 3/20 0.50
CYP2C9 P11712 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
MAPK1 P28482 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
L3MBTL1 Q9Y468 2/20 0.48
KDM4E B2RXH2 1/20 0.48
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4866324 0.87 ALDH1A1 (0.50) CTSBHTTMAPTALDH1A1CYP1A2
SCHEMBL3643443 0.86 CYP1A2 (0.52) CTSBHTTMAPTALDH1A1CYP1A2
SCHEMBL8692030 0.84 SIRT6 (0.52) HTTMAPTALDH1A1CYP1A2LMNA
SCHEMBL24130664 0.83 HTR3A (0.50) MAPTALDH1A1LMNASMN1; SMN2MAPK1
Hydrochloric Acid SCHEMBL30481714 0.82 MAPT (0.51) MAPTALDH1A1LMNASMN1; SMN2MAPK1
SCHEMBL27888685 0.81 CTSB (0.57) CTSBHTTMAPTALDH1A1CYP1A2
SCHEMBL2206983 0.81 CTSB (0.68) CTSBHTTMAPTALDH1A1CYP1A2
SCHEMBL30779614 0.81 CTSB (0.68) CTSBHTTMAPTALDH1A1CYP1A2
SCHEMBL24130778 0.80 HTT (0.53) HTTMAPTALDH1A1CYP1A2LMNA
SCHEMBL11398153 0.79 HTT (0.54) CTSBHTTMAPTALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010125103-A1 DIKETOPIPERAZINE DERIVATIVES AS P2X7 MODULATORS GLAXO GROUP LIMITED (GB) 2010-11-04 WO disclosed