Aurantiogliocladin

Aurantiogliocladin

SCHEMBL487583

COC1=C(OC)C(=O)C(C)=C(C)C1=O

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.50
TDP1 Q9NUW8 4/20 0.50
IDO1 P14902 3/20 0.50
ALDH1A1 P00352 3/20 0.50
LMNA P02545 3/20 0.50
CDC25A P30304 2/20 0.50
CDC25B P30305 2/20 0.50
CYP3A4 P08684 2/20 0.50
CYP2D6 P10635 2/20 0.50
CYP2C9 P11712 2/20 0.50
CYP2C19 P33261 2/20 0.50
KDM4E B2RXH2 2/20 0.50
MAP2K7 O14733 1/20 0.50
GMNN O75496 1/20 0.50
TP53 P04637 1/20 0.50
CYP1A2 P05177 1/20 0.50
POLB P06746 1/20 0.50
HPGD P15428 1/20 0.50
ALOX15 P16050 1/20 0.50
THPO P40225 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12592463 0.88 CDC25A (0.58) MAPTTDP1IDO1ALDH1A1LMNA
SCHEMBL9655485 0.87 CDC25A (0.64) MAPTTDP1IDO1ALDH1A1LMNA
SCHEMBL3420496 0.82 MAPT (0.58) MAPTTDP1IDO1ALDH1A1LMNA
SCHEMBL9180312 0.81 DUSP3 (0.48) MAPTTDP1IDO1ALDH1A1LMNA
SCHEMBL487582 0.81 IDO1 (0.42) MAPTTDP1IDO1ALDH1A1LMNA
SCHEMBL4725792 0.81 APEX1 (0.44) MAPTTDP1IDO1ALDH1A1LMNA
SCHEMBL5158684 0.81 DUSP3 (0.42) MAPTTDP1IDO1ALDH1A1LMNA
SCHEMBL8252760 0.81 AURKA (0.46) MAPTTDP1IDO1ALDH1A1LMNA
SCHEMBL5590298 0.80 CDC25A (0.56) MAPTTDP1IDO1ALDH1A1LMNA
SCHEMBL13033957 0.77 MAPT (0.61) MAPTTDP1IDO1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 72 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080306054-A1 Pharmaceutical Compounds ASTEX THERAPEUTICS LIMITED (GB) 2008-12-11 US claimed
EP-1883402-A2 HYDROXYBENZAMIDE DERIVATIVES AND THEIR USE AS INHIBITORS OF HSP90 Astex Therapeutics Limited (GB) 2008-02-06 EP claimed
WO-2006109075-A2 HYDROXYBENZAMIDE DERIVATIVES AND THEIR USE AS INHIBITORS OF HSP90 ASTEX THERAPEUTICS LIMITED (GB) 2006-10-19 WO claimed
EP-3858351-A1 PHARMACEUTICAL COMPOSITION FOR TREATING FIBROSIS LTT Bio-Pharma Co., Ltd. (JP) 2021-08-04 EP disclosed
US-20210130457-A1 COMPOSITIONS AND METHODS FOR ANTIBODY PRODUCTION IMMUNOGEN, INC 2021-05-06 US disclosed
US-10913795-B2 Compositions and methods for antibody production IMMUNOGEN, INC. (US) 2021-02-09 US disclosed
WO-2019113210-A1 PHOSPHONIUM-BASED IONIC DRUG CONJUGATES ANTHOS PARTNERS, LP (US) 2019-06-13 WO disclosed
US-20190119374-A1 COMPOSITIONS AND METHODS FOR ANTIBODY PRODUCTION IMMUNOGEN, INC. 2019-04-25 US disclosed
EP-2238968-B1 Skin treatment fighting skin aging HENKEL AG & CO KGAA (DE) 2018-05-02 EP disclosed
EP-2841169-B1 HAIR PREPARATIONS COMPRISING HYDROXY-TERMINATED ORGANOPOLYSILOXANE(S) AND THICKENER(S) HENKEL AG & CO KGAA (DE) 2018-04-04 EP disclosed
US-9801922-B2 Compositions and methods of treating cancer UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 2017-10-31 US disclosed
WO-2005019233-A1 MITOQUINONE DERIVATIVES USED AS MITOCHONDRIALLY TARGETED ANTIOXIDANTS ANTIPODEAN PHARMACEUTICALS, INC. (US) 2005-03-03 WO disclosed
EP-1169466-A4 SYNTHESIS OF 1,2,3,4-TETRAHYDROXYBENZENES AND 1,2,3-TRIHYDROXYBENZENES USING MYO-INOSITOL-1-PHOSPHATE SYNTHASE AND MYO-INOSITOL 2-DEHYDROGENASE UNIV MICHIGAN STATE (US) 2005-02-23 EP disclosed
US-20040209337-A1 Synthesis of 1,2,3,4-tetrahydroxybenzenes from biomass-derived carbon NATIONAL SCIENCE FOUNDATION 2004-10-21 US disclosed
US-6750049-B1 Synthesis of 1,2,3,4-tetrahydroxybenzenes and 1,2,3-trihydroxybenzenes using myo-inositol-1-phosphate synthase and myo-inositol 2-dehydrogenase BOARD OF TRUSTEES OPERATING MICHIGAN STATE UNIVERSITY 2004-06-15 US disclosed
US-20030082101-A1 Accelerators for increasing the rate of formation of free radicals and reactive oxygen species CAVALIER DISCOVERY 2003-05-01 US disclosed
WO-2002100478-A9 ACCELERATORS FOR INCREASING THE RATE OF FORMATION OF FREE RADICALS AND REACTIVE OXYGEN SPECIES CAVALIER DISCOVERY (US) 2003-03-27 WO disclosed
WO-2002100478-A2 ACCELERATORS FOR INCREASING THE RATE OF FORMATION OF FREE RADICALS AND REACTIVE OXYGEN SPECIES CAVALIER DISCOVERY (US) 2002-12-19 WO disclosed
EP-1169466-A1 SYNTHESIS OF 1,2,3,4-TETRAHYDROXYBENZENES AND 1,2,3-TRIHYDROXYBENZENES USING MYO-INOSITOL-1-PHOSPHATE SYNTHASE AND MYO-INOSITOL 2-DEHYDROGENASE Board of Trustees operating Michigan State University (US) 2002-01-09 EP disclosed
WO-2000056911-A1 SYNTHESIS OF 1,2,3,4-TETRAHYDROXYBENZENES AND 1,2,3-TRIHYDROXYBENZENES USING MYO-INOSITOL-1-PHOSPHATE SYNTHASE AND MYO-INOSITOL 2-DEHYDROGENASE BOARD OF TRUSTEES OPERATING MICHIGAN STATE UNIVERSITY (US) 2000-09-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030082101-A1 Accelerators for increasing the rate of formation of free radicals and reactive oxygen species SOD1, SOD3, APEX1 MAPT 3245/4885TDP1 697/4885IDO1 2808/4885
US-20190119374-A1 COMPOSITIONS AND METHODS FOR ANTIBODY PRODUCTION TXNRD1, P4HB, CYBB MAPT 3936/4885TDP1 4634/4885IDO1 2753/4885
US-10913795-B2 Compositions and methods for antibody production TXNRD1, P4HB, CYBB MAPT 3936/4885TDP1 4634/4885IDO1 2753/4885
US-20080306054-A1 Pharmaceutical Compounds HSP90AB1, HSP90AA1, HSP90AB2P MAPT 82/4885TDP1 1397/4885IDO1 853/4885
US-20210130457-A1 COMPOSITIONS AND METHODS FOR ANTIBODY PRODUCTION TXNRD1, P4HB, CYBB MAPT 3936/4885TDP1 4634/4885IDO1 2753/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.