SCHEMBL4886491

SCHEMBL4886491

Cc1cc(C23CC4CC(CC(C4)C2)C3)c(O)c(S(=O)(=O)Nc2ccc(C#N)cc2Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 2/20 0.45
ACLY P53396 4/20 0.40
PGR P06401 1/20 0.39
HSD11B1 P28845 2/20 0.39
MAPK1 P28482 1/20 0.36
PDK1 Q15118 1/20 0.36
PDK2 Q15119 1/20 0.36
PDK3 Q15120 1/20 0.36
PDK4 Q16654 1/20 0.36
PIK3C3 Q8NEB9 1/20 0.35
WDR5 P61964 1/20 0.35
GPR119 Q8TDV5 3/20 0.34
ATM Q13315 1/20 0.34
CNR2 P34972 1/20 0.34
STS P08842 1/20 0.33
TSHR P16473 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4897237 0.89 SLC22A12 (0.45) SLC22A12ACLYPGRHSD11B1WDR5
SCHEMBL4886499 0.88 ACLY (0.44) SLC22A12ACLYPGRHSD11B1PDK1
SCHEMBL4884915 0.85 PGR (0.52) SLC22A12PGRTSHR
SCHEMBL4897107 0.82 CRHBP (0.46) MAPK1NPSR1
SCHEMBL4893835 0.79 SLC22A12 (0.57) SLC22A12ACLYMAPK1PDK1PDK2
SCHEMBL4895380 0.73 PGR (0.49) SLC22A12PGRWDR5
SCHEMBL4896573 0.73 PGR (0.49) SLC22A12PGRTSHR
SCHEMBL4890237 0.72 MEN1 (0.33) MAPK1CNR2
SCHEMBL4898138 0.70 SLC22A12 (0.57) SLC22A12ACLYHSD11B1PDK1PDK2
SCHEMBL4895370 0.70 KDM4E (0.41) MAPK1CNR2STS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080255240-A1 Sulfonamide Derivatives NOVO NORDISK A/S (DK) 2008-10-16 US claimed
EP-1756025-A1 SULFONAMIDE DERIVATIVES NOVO NORDISK A/S (DK) 2007-02-28 EP claimed
WO-2005105712-A1 SULFONAMIDE DERIVATIVES NOVO NORDISK A/S (DK) 2005-11-10 WO claimed
US-20080255240-A1 Sulfonamide Derivatives NOVO NORDISK A/S (DK) 2008-10-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080255240-A1 Sulfonamide Derivatives FABP4, SQOR, CS SLC22A12 1558/4885ACLY 167/4885PGR 4193/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.