Elisartan

Elisartan

SCHEMBL489079

CCCCc1nc(Cl)c(C(=O)OC(C)OC(=O)OCC)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 3/20 0.53
AGTR2 P50052 3/20 0.53
PPARG P37231 1/20 0.45
KCNH2 Q12809 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Elisartan SCHEMBL489081 1.00 AGTR1 (0.53) AGTR1AGTR2PPARGKCNH2
Elisartan SCHEMBL29595840 0.99 AGTR1 (0.52) AGTR1AGTR2PPARGKCNH2
Elisartan SCHEMBL1560942 0.99 AGTR1 (0.52) AGTR1AGTR2PPARGKCNH2
Elisartan SCHEMBL615371 0.99 AGTR1 (0.52) AGTR1AGTR2PPARGKCNH2
Elisartan SCHEMBL615370 0.99 AGTR1 (0.52) AGTR1AGTR2PPARGKCNH2
SCHEMBL12990879 0.93 AGTR2 (0.53) AGTR1AGTR2PPARG
SCHEMBL6130076 0.92 AGTR1 (0.48) AGTR1AGTR2
SCHEMBL4609266 0.92 AGTR1 (0.48) AGTR1AGTR2
SCHEMBL12991717 0.91 AGTR2 (0.51) AGTR1AGTR2
SCHEMBL13771416 0.91 AGTR1 (0.48) AGTR1AGTR2PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 836 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250082608-A1 TREATMENT AND PREVENTION OF GLOMERULAR DISEASE SINGAPORE HEALTH SERVICES PTE LTD. (SG) 2025-03-13 US claimed
EP-4448096-A1 TREATMENT AND PREVENTION OF GLOMERULAR DISEASE Singapore Health Services Pte. Ltd. (SG) 2024-10-23 EP claimed
EP-3873904-B1 TETRAHYDROPYRAN (THP)-SUBSTITUTED BICYCLIC-PYRIMIDINEDIONE COMPOUNDS MYOKARDIA INC (US) 2024-07-10 EP claimed
US-12016835-B2 Neprilysin inhibitors THERAVANCE BIOPHARMA R&D IP, LLC (US) 2024-06-25 US claimed
US-11851443-B2 Neprilysin inhibitors THERAVANCE BIOPHARMA R&D IP, LLC (US) 2023-12-26 US claimed
US-20230285340-A1 NEPRILYSIN INHIBITORS THERAVANCE BIOPHARMA R&D IP LLC (US) 2023-09-14 US claimed
US-11718591-B2 Crystalline (2S,4R)-5-(5′-chloro-2′-fluoro-[1,1′-biphenyl]-4-yl)-2-(ethoxymethyl)-4-(3-hydroxyisoxazole-5-carboxamido)-2- methylpentanoic acid and uses thereof THERAVANCE BIOPHARMA R&D IP, LLC (US) 2023-08-08 US claimed
WO-2023111196-A1 TREATMENT AND PREVENTION OF GLOMERULAR DISEASE SINGAPORE HEALTH SERVICES PTE. LTD. (SG) 2023-06-22 WO claimed
US-11634413-B2 Neprilysin inhibitors THERAVANCE BIOPHARMA R&D IP, LLC (US) 2023-04-25 US claimed
US-20220340569-A1 SUBSTITUTED 5,6,7,8-TETRAHYDROPYRIDO[2,3-D]PYRIMIDINE-2,4-DIONES FOR TREATING CARDIAC DISEASES MYOKARDIA INC (US) 2022-10-27 US claimed
EP-1545540-A2 COMBINATION THERAPY USING A DUAL PPAR ALPHA/GAMMA AGONIST AND AN ANGIOTENSIN II TYPE I RECEPTOR ANTAGONIST Merck & Co., Inc. (US) 2005-06-29 EP claimed
WO-2005023182-A2 NITROSATED AND NITROSYLATED CARDIOVASCULAR COMPOUNDS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2005-03-17 WO claimed
WO-2004017896-A2 COMBINATION THERAPY USING A DUAL PPAR ALPHA/GAMMA AGONIST AND AN ANGIOTENSIN II TYPE I RECEPTOR ANTAGONIST MERCK & CO., INC. (US) 2004-03-04 WO claimed
EP-1393722-A2 Use of angiotensin II subtype 1 (AT1) antagonists for the manufacture of a medicament in the treatment of premenstrual syndrome DePadova, Anthony S. (US) 2004-03-03 EP claimed
US-6653306-B1 Circulatory disorders G.D. SEARLE & CO. 2003-11-25 US claimed
EP-0831911-B1 SPIRONOLACTONE AND ANGIOTENSIN II ANTAGONIST COMBINATION THERAPY FOR TREATMENT OF CONGESTIVE HEART FAILURE SEARLE & CO (US) 2002-04-17 EP claimed
EP-0759754-A4 A METHOD OF MODIFYING ANGIOTENSIN RECEPTOR ACTIVITY FOR TREATMENT OF PREMENSTRUAL SYNDROME AND MEDIATION OF PAIN DEPADOVA ANTHONY S (US) 2000-07-05 EP claimed
US-5753651-A Use of AT1 antagonist such as irbesartan or candesartan cilexetil, among others; premenstrual syndrome (PMS) DEPADOVA ANTHONY S (US) 1998-05-19 US claimed
EP-0759754-A1 A METHOD OF MODIFYING ANGIOTENSIN RECEPTOR ACTIVITY FOR TREATMENT OF PREMENSTRUAL SYNDROME AND MEDIATION OF PAIN DePadova, Anthony S. (US) 1997-03-05 EP claimed
WO-1995029674-A1 A METHOD OF MODIFYING ANGIOTENSIN RECEPTOR ACTIVITY FOR TREATMENT OF PREMENSTRUAL SYNDROME AND MEDIATION OF PAIN DEPADOVA ANTHONY S (US) 1995-11-09 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230285340-A1 NEPRILYSIN INHIBITORS MME, REN, ACE AGTR1 5/4885AGTR2 11/4885PPARG 4731/4885
US-11718591-B2 Crystalline (2S,4R)-5-(5′-chloro-2′-fluoro-[1,1′-biphenyl]-4-yl)-2-(ethoxymethyl)-4-(3-hydroxyisoxazole-5-carboxamido)-2- methylpentanoic acid and uses thereof MME, CTSC, REN AGTR1 25/4885AGTR2 42/4885PPARG 3055/4885
US-20220340569-A1 SUBSTITUTED 5,6,7,8-TETRAHYDROPYRIDO[2,3-D]PYRIMIDINE-2,4-DIONES FOR TREATING CARDIAC DISEASES DHPS, THPO, TNNI3 AGTR1 1015/4885AGTR2 868/4885PPARG 876/4885
US-11634413-B2 Neprilysin inhibitors MME, REN, ACE AGTR1 4/4885AGTR2 13/4885PPARG 4587/4885
US-11851443-B2 Neprilysin inhibitors MME, REN, ACE AGTR1 4/4885AGTR2 9/4885PPARG 4814/4885
US-12016835-B2 Neprilysin inhibitors MME, REN, ACE AGTR1 5/4885AGTR2 11/4885PPARG 4731/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.