SCHEMBL490315

SCHEMBL490315

NS(=O)(=O)N1CCOCC1

nearest known ligand 0.65

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.65
CA7 P43166 2/20 0.65
CA14 Q9ULX7 1/20 0.65
SMN1; SMN2 Q16637 4/20 0.54
TSHR P16473 3/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
CA1 P00915 3/20 0.52
CA2 P00918 3/20 0.52
POLB P06746 3/20 0.45
LMNA P02545 1/20 0.41
CA13 Q8N1Q1 1/20 0.41
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL29968774 0.97 CA12 (0.62) CA12CA7CA14SMN1; SMN2TSHR
SCHEMBL28233992 0.92 SMN1; SMN2 (0.67) CA12CA7CA14SMN1; SMN2TSHR
SCHEMBL23592712 0.90 SMN1; SMN2 (0.58) CA12CA7CA14SMN1; SMN2TSHR
SCHEMBL5473926 0.83
SCHEMBL4724826 0.79 CA12 (1.00) CA12CA7CA14SMN1; SMN2TSHR
SCHEMBL4141702 0.77
SCHEMBL11688163 0.77 CA1 (0.69) CA12CA7CA14SMN1; SMN2TSHR
SCHEMBL222875 0.77 CA12 (0.65) CA12CA7CA14SMN1; SMN2TSHR
SCHEMBL898965 0.77 CA12 (0.65) CA12CA7CA14SMN1; SMN2TSHR
SCHEMBL995945 0.74 CA12 (0.62) CA12CA7CA14SMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 804 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4192833-B1 PHARMACOLOGICALLY ACTIVE HETEROCYCLIC-SUBSTITUTED PYRAZOLO[1,5-A]PYRIMIDINE DERIVATIVES RICHTER GEDEON NYRT (HU) 2026-01-21 EP claimed
CN-118666780-A Method for preparing morpholinosulfonamide compound by microwave promotion 邵阳学院 2024-09-20 CN claimed
CN-117384673-A Extraction process for producing heavy aromatic derivative 宁波博汇化工科技股份有限公司 2024-01-12 CN claimed
EP-3860998-B1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH APJ RECEPTOR ACTIVITY ANNAPURNA BIO INC (US) 2023-12-27 EP claimed
US-11471455-B2 Compounds and compositions for treating conditions associated with APJ receptor activity ANNAPURNA BIO, INC. (US) 2022-10-18 US claimed
EP-2350068-B1 UREA DERIVATIVES OF SUBSTITUTED NORTROPANES, MEDICAMENTS CONTAINING SUCH COMPOUNDS AND THEIR USE BOEHRINGER INGELHEIM INT (DE) 2017-08-30 EP claimed
CN-103339132-B Purinylpyridinylamino-2,4-difluorophenyl sulfonamide derivative, pharmaceutically acceptable salt thereof, preparation method thereof, and pharmaceutical composition with inhibitory activity against raf kinase, containing same as active ingredi 株式会社麦迪帕克特 2017-02-15 CN claimed
EP-2863914-A1 PYRAZOLYL DERIVATIVES AS SYK INHIBITORS Merck Sharp & Dohme Corp. (US) 2015-04-29 EP claimed
WO-2013192125-A1 PYRAZOLYL DERIVATIVES AS SYK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2013-12-27 WO claimed
CN-103339132-A Novel purinylpyridinylamino-2,4-difluorophenyl sulfonamide derivative, pharmaceutically acceptable salt thereof, preparation method thereof, and pharmaceutical composition with inhibitory activity against raf kinase, containing same as active ingredi YOUAI CO LTD 2013-10-02 CN claimed
US-20040048880-A1 Bicyclic heterocyclic compounds, pharmaceutical compositions containing these compounds, their use and process for preparing them BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2004-03-11 US claimed
EP-0637965-B1 ENHANCED TRIPLE-HELIX AND DOUBLE-HELIX FORMATION WITH OLIGOMERS CONTAINING MODIFIED PYRIMIDINES ISIS PHARMACEUTICALS INC (US) 2002-10-16 EP claimed
US-20020128247-A1 Beta3 agonists and uses thereof DOW ROBERT L (US) 2002-09-12 US claimed
EP-1236723-A1 Sulfamide derivatives useful as beta3 agonists and pharmaceutical uses thereof Pfizer Products Inc. (US) 2002-09-04 EP claimed
WO-2001040515-A1 GAPPED OLIGOMERS HAVING SITE SPECIFIC CHIRAL PHOSPHOROTHIOATE INTERNUCLEOSIDE LINKAGES ISIS PHARMACEUTICALS, INC. (US) 2001-06-07 WO claimed
US-5843905-A Peptidic phosphinyloxymethyl ketones as interleukin-1β-converting enzyme inhibitors VERTEX PHARMACEUTICALS, INCORPORATED (US) 1998-12-01 US claimed
EP-0644197-B1 Peptidic phosphinyloxymethyl ketones as interleukin-1beta-converting enzyme inhibitors VERTEX PHARMA (US) 1998-09-09 EP claimed
US-5677283-A α-heteroaryloxymethyl ketones as interleukin - 1 β converting enzyme inhibitors SANOFI (FR) 1997-10-14 US claimed
EP-0644198-A1 Alpha-heteroaryloxymethyl ketones as interleukin-1beta converting enzyme inhibitors STERLING WINTHROP INC. (US) 1995-03-22 EP claimed
EP-0644197-A1 Peptidic phosphinyloxymethyl ketones as interleukin-1beta-converting enzyme inhibitors STERLING WINTHROP INC. (US) 1995-03-22 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020128247-A1 Beta3 agonists and uses thereof ADRB3, ADRB1, ADRB2 CA12 4686/4885CA7 4193/4885CA14 4779/4885
US-11471455-B2 Compounds and compositions for treating conditions associated with APJ receptor activity APLNR, AGTR1, AGTR2 CA12 2101/4885CA7 2242/4885CA14 3885/4885
US-20040048880-A1 Bicyclic heterocyclic compounds, pharmaceutical compositions containing these compounds, their use and process for preparing them CYP11B1, AR, CYP11B2 CA12 1870/4885CA7 1390/4885CA14 2174/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.