SCHEMBL4904285

SCHEMBL4904285

COC(=O)c1cc(S(=O)(=O)N(CCc2ccc(OCc3ccc(F)c(F)c3)cc2)Cc2ccc(F)c(F)c2)ccc1C

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.45
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
LMNA P02545 2/20 0.42
TAS2R14 Q9NYV8 3/20 0.42
MAPT P10636 1/20 0.42
BMP1 P13497 3/20 0.42
CA12 O43570 4/20 0.41
CA1 P00915 4/20 0.41
CA2 P00918 4/20 0.41
CA4 P22748 4/20 0.41
CA9 Q16790 4/20 0.41
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4897933 0.91 TAS2R14 (0.46) MAOAMAOBLMNATAS2R14MAPT
SCHEMBL4900038 0.89 TAS2R14 (0.46) TP53LMNATAS2R14MAPTBMP1
SCHEMBL4904145 0.89 MMP2 (0.45) TP53LMNATAS2R14MAPTBMP1
SCHEMBL4902732 0.88 KMT2A (0.48) TP53TAS2R14BMP1CA12CA1
SCHEMBL4908413 0.87 CNR2 (0.48) TP53LMNATAS2R14MAPTBMP1
SCHEMBL4895626 0.86 TAS2R14 (0.56) TP53LMNATAS2R14MAPTBMP1
SCHEMBL4905637 0.86 TAS2R14 (0.44) TP53LMNATAS2R14MAPTBMP1
SCHEMBL4905982 0.85 BMP1 (0.49) MAOBTAS2R14MAPTBMP1CA12
Methane SCHEMBL6506917 0.84 BMP1 (0.48) MAOBTAS2R14MAPTBMP1CA12
SCHEMBL4895596 0.83 LMNA (0.42) TP53LMNATAS2R14BMP1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080090829-A1 SUBSTITUTED HETEROARYL- AND PHENYLSULFAMOYL COMPOUNDS PFIZER INC. 2008-04-17 US disclosed
US-20080090829-A1 SUBSTITUTED HETEROARYL- AND PHENYLSULFAMOYL COMPOUNDS PFIZER INC. 2008-04-17 US disclosed
US-20080090829-A1 SUBSTITUTED HETEROARYL- AND PHENYLSULFAMOYL COMPOUNDS PFIZER INC. 2008-04-17 US disclosed
US-20060229363-A1 Substituted Heteroaryl- and Phenylsulfamoyl Compounds HAMANAKA ERNEST S 2006-10-12 US disclosed
US-20050288340-A1 Substituted heteroaryl- and phenylsulfamoyl compounds PFIZER INC 2005-12-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060229363-A1 Substituted Heteroaryl- and Phenylsulfamoyl Compounds PPARA, PPARG, PPARD TP53 3260/4885MAOA 4248/4885MAOB 4126/4885
US-20050288340-A1 Substituted heteroaryl- and phenylsulfamoyl compounds PPARA, PPARG, PPARD TP53 3421/4885MAOA 4248/4885MAOB 4263/4885
US-20080090829-A1 SUBSTITUTED HETEROARYL- AND PHENYLSULFAMOYL COMPOUNDS PPARA, PPARG, PPARD TP53 3421/4885MAOA 4248/4885MAOB 4263/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.