SCHEMBL490769

SCHEMBL490769

CCOC(=O)C(Cc1ccc(O)c(OC)c1)C(=O)OCC

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B2 P37059 2/20 0.60
FOS P01100 1/20 0.60
TTR P02766 1/20 0.60
JUN P05412 1/20 0.60
NR3C1 P04150 1/20 0.60
HSD17B1 P14061 1/20 0.60
MMP1 P03956 1/20 0.57
CYP3A4 P08684 1/20 0.57
ALOX15 P16050 1/20 0.56
ALOX12 P18054 1/20 0.56
ALDH1A1 P00352 2/20 0.55
TSHR P16473 2/20 0.55
GAA P10253 1/20 0.55
NFKB1 P19838 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
LDHA P00338 1/20 0.55
ALOX5 P09917 1/20 0.51
OR51E2 Q9H255 1/20 0.51
KDM4E B2RXH2 1/20 0.51
TAAR1 Q96RJ0 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL933495 0.96 HSD17B2 (0.56) HSD17B2FOSTTRJUNNR3C1
SCHEMBL935389 0.92 HSD17B2 (0.56) HSD17B2FOSTTRJUNNR3C1
SCHEMBL934179 0.91 HSD17B2 (0.51) HSD17B2FOSTTRJUNNR3C1
SCHEMBL490506 0.88 ALOX15 (0.60) CYP3A4ALOX15ALOX12TSHRGAA
SCHEMBL491026 0.88 LDHA (0.71) ALOX15ALOX12ALDH1A1GAALDHA
SCHEMBL934471 0.88 FOS (0.64) HSD17B2FOSTTRJUNNR3C1
SCHEMBL5685173 0.87 HSD17B2 (0.63) HSD17B2FOSTTRJUNNR3C1
SCHEMBL5685443 0.87 HSD17B2 (0.59) HSD17B2FOSTTRJUNNR3C1
SCHEMBL5382445 0.86 HSD17B2 (0.57) HSD17B2FOSTTRJUNNR3C1
SCHEMBL933400 0.86 FOS (0.61) HSD17B2FOSTTRJUNNR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011006566-A2 MONOMETHOXY-HYDROXY-BENZYLMALONATES MERCK PATENT GMBH (DE) 2011-01-20 WO claimed
EP-2238964-A2 Stabilised cosmetic compounds Henkel AG & Co. KGaA (DE) 2010-10-13 EP claimed
US-8268293-B2 Using compounds which do not themselves exhibit significant UV absorption in the UV-A or UV-B region, but are reactive under use conditions, such as 4-hydroxyphenylpropionic acid, or 2-ethylhexyl 4-hydroxy-3,5-dimethoxycinnamate, or polysiloxanes which contain benzylidenemalonic acid derivatives MERCK PATENT GMBH (DE) 2012-09-18 US disclosed
US-8106233-B2 Applying di-2-ethylhexyl 4-hydroxy-3,5-dimethoxy-benzylmalonate; protective action against UV rays, oxidative stress on body cells, counters skin ageing MERCK PATENT GMBH (DE) 2012-01-31 US disclosed
WO-2011006566-A2 MONOMETHOXY-HYDROXY-BENZYLMALONATES MERCK PATENT GMBH (DE) 2011-01-20 WO disclosed
WO-2011006566-A2 MONOMETHOXY-HYDROXY-BENZYLMALONATES MERCK PATENT GMBH (DE) 2011-01-20 WO disclosed
EP-2238964-A2 Stabilised cosmetic compounds Henkel AG & Co. KGaA (DE) 2010-10-13 EP disclosed
US-20080171004-A1 Using compounds which do not themselves exhibit significant UV absorption in the UV-A or UV-B region, but are reactive under use conditions, such as 4-hydroxyphenylpropionic acid, or 2-ethylhexyl 4-hydroxy-3,5-dimethoxycinnamate, or polysiloxanes which contain benzylidenemalonic acid derivatives MERCK PATENT GMBH (DE) 2008-07-17 US disclosed
US-20080152603-A1 Antioxidants SUSONITY Commercial GmbH (DE) 2008-06-26 US disclosed
CN-101163659-A Antioxidants MERCK PATENT GMBH (DE) 2008-04-16 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080152603-A1 Antioxidants GPX4, GPX1, CAT HSD17B2 684/4885FOS 647/4885TTR 423/4885
US-20080171004-A1 Using compounds which do not themselves exhibit significant UV absorption in the UV-A or UV-B region, but are reactive under use conditions, such as 4-hydroxyphenylpropionic acid, or 2-ethylhexyl 4-hydroxy-3,5-dimethoxycinnamate, or polysiloxanes which contain benzylidenemalonic acid derivatives HPD, HAAO, UGT1A6 HSD17B2 953/4885FOS 1552/4885TTR 3973/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.