SCHEMBL4909466

SCHEMBL4909466

CCC(C)(Oc1ccccc1)S(=O)(=O)NC

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 2/20 0.36
NPSR1 Q6W5P4 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HTT P42858 2/20 0.34
LMNA P02545 1/20 0.34
PPARA Q07869 2/20 0.34
MMP1 P03956 3/20 0.33
MMP13 P45452 3/20 0.33
MMP2 P08253 2/20 0.33
ALDH1A1 P00352 1/20 0.33
PGR P06401 1/20 0.33
CYP2C19 P33261 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HTR1D P28221 1/20 0.33
HTR1B P28222 1/20 0.33
PSIP1 O75475 1/20 0.33
PPARG P37231 1/20 0.33
MMP9 P14780 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6238670 0.79 CA1 (0.42) NPSR1HTTLMNAMMP1MMP13
SCHEMBL4909452 0.71 ALDH1A1 (0.37) NR3C2NPSR1HTTLMNAMMP1
SCHEMBL9541482 0.70 PPARG (0.39) NPSR1L3MBTL1PPARAPPARG
SCHEMBL3081094 0.68 LTA4H (0.40) NPSR1L3MBTL1LMNAPPARACYP2C19
SCHEMBL183720 0.68 LTA4H (0.40) NPSR1L3MBTL1PPARAALDH1A1PPARG
SCHEMBL1453725 0.68 LTA4H (0.40) NPSR1L3MBTL1PPARACYP2C19PPARG
SCHEMBL4904737 0.67 PPARG (0.47) NPSR1L3MBTL1PPARAPPARG
SCHEMBL8397511 0.66 CA1 (0.47) NR3C2NPSR1L3MBTL1HTTLMNA
SCHEMBL5286690 0.65 TAAR1 (0.40) NPSR1L3MBTL1PPARAALDH1A1PPARG
SCHEMBL13363806 0.65 LTA4H (0.38) NPSR1L3MBTL1PPARAPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200352946-A1 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASES RESVERLOGIX CORP. 2020-11-12 US disclosed
US-20180104245-A1 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASES HEPALINK (HONG KONG) LIMITED (HK) 2018-04-19 US disclosed
US-20160106750-A1 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASES RESVERLOGIX CORP. (CA) 2016-04-21 US disclosed
US-9199990-B2 Compounds for the prevention and treatment of cardiovascular diseases RESVERLOGIX CORP. (CA) 2015-12-01 US disclosed
US-20150072955-A1 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASES RESVERLOGIX CORP. (US) 2015-03-12 US disclosed
US-8889698-B2 Compounds for the prevention and treatment of cardiovascular diseases RESVERLOGIX CORP. (CA) 2014-11-18 US disclosed
US-20080188467-A1 To regulate the expression of apolipoprotein A-I; atherosclerosis; improved pharmacological properties; 3-(4-hydroxy-3,5-dimethylphenyl)-6,8-dimethoxyisoquinolin-1(2H)-one; to reduce cholesterol levels; agonists HEPALINK (HONG KONG) LIMITED (HK) 2008-08-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180104245-A1 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASES APOB, HDLBP, FABP3 NR3C2 946/4885NPSR1 2771/4885L3MBTL1 1494/4885
US-20200352946-A1 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASES APOB, HDLBP, FABP3 NR3C2 946/4885NPSR1 2771/4885L3MBTL1 1494/4885
US-20160106750-A1 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASES APOB, HDLBP, FABP3 NR3C2 946/4885NPSR1 2771/4885L3MBTL1 1494/4885
US-20150072955-A1 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASES APOB, HDLBP, FABP3 NR3C2 946/4885NPSR1 2771/4885L3MBTL1 1494/4885
US-20080188467-A1 To regulate the expression of apolipoprotein A-I; atherosclerosis; improved pharmacological properties; 3-(4-hydroxy-3,5-dimethylphenyl)-6,8-dimethoxyisoquinolin-1(2H)-one; to reduce cholesterol levels; agonists APOB, LDLR, APOL1 NR3C2 449/4885NPSR1 1997/4885L3MBTL1 2366/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.